热门产品推荐HOT PRODUCTS
- Doxorubicin
Doxorubicin (Adriamycin)是一种抗生素类试剂,能够抑制DNA拓扑异构酶II,且诱导DNA损伤和凋亡。
- N6-methyladenosine
N6-methyladenosine (m6A)是碱基修饰的腺苷类似物,在天然RNAs中作为稀有核苷。N6-methyladenosine(m6A)是mRNA的第五种碱基。
- Doxycycline HCl
Doxycycline盐酸盐是合成的四环素类衍生物,具有抗菌活性。
- SB216763
SB216763, a potent and selective cell permeable GSK-3 inhibitor, is equally effective at inhibiting human GSK-3α and GSK-3β. SB216763是一种有效的,选择...
- Tacrolimus
Tacrolimus (FK506)是一种免疫抑制剂和大环内酯类抗生素,用于同种异体的器官移植,可以降低病人的免疫系统的作用。
- Go6976
Go6976 is a potent protein kinase C (PKC) inhibitor (IC50 = 7.9 nM), selectively inhibits PKCα, and PKCβ1 (IC50 values are 2.3 and 6.2 nM respectively...
- TAK-875
TAK-875是一种选择性GPR40激动剂,EC50为14 nM,比油酸有效400倍。
- Docetaxel
Docetaxel, a cytotoxic antimicrotuble agent, is frequently administrated as a first line treatment for prostate cancers. Docetaxel,一种紫杉醇类似物,通...
- Enzalutamide
Enzalutamide, an AR signaling inhibitor, is effective for bicalutamide-resistant tumors and has been used in metastatic castration-resistant prostate ...
- SP600125
SP600125是一种广谱JNK抑制剂,作用于JNK1, JNK2和JNK3时,IC50分别为40 nM, 40 nM和90 nM,比作用于MKK4选择性高10倍,比作用于MKK3, MKK6, PKB,和PKCα选择性高25倍...
- Rapamycin
Rapamycin, an mTOR inhibitor, shows potent immunosuppressive and antiproliferative properties. Rapamycin是一种常用的选择性的mTOR抑制剂,IC50为~0.1 nM。
- Lapatinib
Lapatinib (GW572016) is a small-molecule dual inhibitor of EGFR and ErbB2 receptor kinase activities. Lapatinib可形成Lapatinib的二甲苯磺酸盐,是一种有效...
- Ibrutinib
Ibrutinib (PCI-32765)是一种有效的,高选择性的Btk抑制剂,IC50为0.5 nM,能稍许微抑制Bmx, CSK, FGR, BRK及HCK,但对EGFR, Yes, ErbB2, JAK3等作用效果稍弱。
- SAHA
Vorinostat (SAHA, MK0683)是一种I和II类组蛋白去乙酰化酶(HDAC)抑制剂,IC50小于86 nM。
- MG-132
MG-132是一种蛋白酶体抑制剂,IC50为100 nM。还能抑制钙蛋白酶,IC50为1.2 μM。