LPA Receptor
LPARs (lysophosphatidic acid receptors) are a group of G protein-coupled receptors for lysophosphatidic acid (LPA) that include:
Lysophosphatidic acid receptor 1 (LPAR1; formerly known as EDG2, GPR26)
Lysophosphatidic acid receptor 2 (LPAR2; formerly known as EDG4)
Lysophosphatidic acid receptor 3 (LPAR3; formerly known as EDG7)
Lysophosphatidic acid receptor 4 (LPAR4; formerly known as GPR23, P2RY9)
Lysophosphatidic acid receptor 5 (LPAR5; formerly known as GPR92)
Lysophosphatidic acid receptor 6 (LPAR6; formerly known as GPR87, P2RY5).
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AM966是高亲和性的口服的溶血磷脂酸（LPA1）受体拮抗剂(IC50=17 nM)，比对其它LPA受体的抑制性高。
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H2L 5765834是LPA1，3，5 拮抗剂。
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H2L5186303是活性的，选择性 LPA2 受体拮抗剂。
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GRI 977143是选择性 LPA2 受体 非lipid 激动剂。
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1-Oleoyl lysophosphatidic acid sodium salt是LPA1 和 LPA2的内源性激动剂。
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