CaMK is an abbreviation for the Ca2+/calmodulin-dependent protein kinase class of enzymes. CAMKs are activated by increases in the concentration of intracellular calcium ions (Ca2+) and transfers phosphates from ATP to defined serine or threonine residues in other proteins. Activated CAMK is involved in the phosphorylation of transcription factors and therefore, in the regulation of expression of responding genes. Members of this enzyme class include: CAMKI(CAMKIα,CAMKIβ,CAMKIδ,CAMKIγ),CAMKII(CAMKIIα,CAMKIIβ,CAMKIIδ,CAMKIIγ,CAMKIII,CAMKIV).
  • Arcyriaflavin A EI0478

    Arcyriaflavin A是活性的cdk4/cyclin D1,CaM 激酶 II 抑制剂。(anti-HCMV)。

  • A 484954 EI0329

    A 484954是CaM 激酶 III (eEF-2 激酶) 抑制剂。

  • STO-609 acetate EI2638

    STO-609 acetate是STO-609 acetate是CaM-KK的抑制剂具有高活性的竞争型选择性特点,并且可以透过细胞膜。

  • KN-62 EY1183

    KN-62 is a selective, cell permeable inhibitor of calcium/calmodulin-dependent kinase II (CaMKII; IC50 = 900 nM).

  • KN-93 Phosphate EY0552

    KN-93 H3PO4 是一种强效的特异性的Ca2+/calmodulin-dependent protein kinase II (CaMKII)抑制剂,其 Ki 为 0.37 μM,对 APK, PKC, MLCK 或 Ca2+-PDE 没有明显的抑制活性。

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