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Melatonin Receptor


Melatonin receptor is a G protein-coupled receptor (GPCR) which binds melatonin. Three types of melatonin receptor have been cloned. The MT1 (or Mel1A or MTNR1A) and MT2 (or Mel1B or MTNR1B) receptor subtypes are present in humans and other mammals, while an additional melatonin receptor subtype MT3 (or Mel1C or MTNR1C) has been identified in amphibia and birds.
  • GR 135531 EI1218

    GR 135531是高亲和性 melatonin MT3 配体。

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  • 6-Chloromelatonin EI0299

    6-Chloromelatonin是Melatonin 激动剂。

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  • 4-P-PDOT EI0286

    4-P-PDOT是MT2 拮抗剂。

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  • 2-Phenylmelatonin EI0254

    2-Phenylmelatonin是活性的 melatonin 激动剂。

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  • 2-Iodomelatonin EI0246

    2-Iodomelatonin是高亲和性 melatonin 激动剂。

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  • GR 135531 EI1218

    GR 135531是高亲和性 melatonin MT3 配体。

    More
  • 6-Chloromelatonin EI0299

    6-Chloromelatonin是Melatonin 激动剂。

    More
  • 4-P-PDOT EI0286

    4-P-PDOT是MT2 拮抗剂。

    More
  • 2-Phenylmelatonin EI0254

    2-Phenylmelatonin是活性的 melatonin 激动剂。

    More
  • 2-Iodomelatonin EI0246

    2-Iodomelatonin是高亲和性 melatonin 激动剂。

    More
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