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CGRP Receptor


Calcitonin gene-related peptide (CGRP) receptor antagonists are a class of drugs that act as antagonists of the calcitonin gene-related peptide receptor (CGRPR). CGRPR antagonists are under investigation as potential antimigraine agents and also in the context of osteoarthritis.

  • MK-3207 HCl EY1485

    MK-3207 HCl是一种有效的CGRP受体拮抗剂，IC50和Ki分别为0.12 nM和0.022 nM，对人AM1， AM2， CTR，和AMY3具有高度选择性。

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