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Vasopressin Receptor


The actions of vasopressin are mediated by stimulation of tissue-specific G protein-coupled receptors (GPCRs) called vasopressin receptors that are classified into V1, V2 and V3 subtypes. These three subtypes differ in localization, function and signal transduction mechanisms.

  • RG7713 EY4823

    RG7713 is a highly potent and selective Brain-Penetrant Vasopressin 1a (V1a) receptor antagonist with Kis of 1 nM (hV1a) and 39 nM (mV1a).

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  • Tolvaptan EY2414

    Tolvaptan is a selective, competitive arginine vasopressin receptor 2 antagonist with an IC50 of 1.28μM for the inhibition of AVP-induced platelet aggregation.

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  • Conivaptan HCl EY2364

    Conivaptan is a non-peptide inhibitor of antidiuretic hormone (vasopressin receptor antagonist).

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