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5-HT Receptor


5-HT receptors (5-hydroxytryptamine receptors,The serotonin receptors) are a group of G protein-coupled receptors (GPCRs) and ligand-gated ion channels (LGICs) found in the central and peripheral nervous systems. They mediate both excitatory and inhibitory neurotransmission. The serotonin receptors are activated by the neurotransmitter serotonin, which acts as their natural ligand.

  • Pimavanserin EY2762

    Pimavanserin is a potent and selective serotonin 5-HT2A inverse agonist with pIC50 of 8.73, used to treat psychosis associated with Parkinson’s disease.

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  • Cyproheptadine hydrochloride EY2718

    Cyproheptadine hydrochloride sesquihydrate is an antihistamine and is an antagonist of serotonin and histamine2.

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  • Trimipramine Maleate EY2633

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  • Cyclobenzaprine HCl EY2586

    Cyclobenzaprine HCl is a muscle relaxant by blocking pain sensations, used for the treatment of muscle spasms.

    More
  • Azacyclonol EY2468

    Azacyclonol, also known as γ-pipradol, is a drug used to diminish hallucinations in psychotic individuals.

    More
  • Pimavanserin EY2762

    Pimavanserin is a potent and selective serotonin 5-HT2A inverse agonist with pIC50 of 8.73, used to treat psychosis associated with Parkinson’s disease.

    More
  • Cyproheptadine hydrochloride EY2718

    Cyproheptadine hydrochloride sesquihydrate is an antihistamine and is an antagonist of serotonin and histamine2.

    More
  • Trimipramine Maleate EY2633

    More
  • Cyclobenzaprine HCl EY2586

    Cyclobenzaprine HCl is a muscle relaxant by blocking pain sensations, used for the treatment of muscle spasms.

    More
  • Azacyclonol EY2468

    Azacyclonol, also known as γ-pipradol, is a drug used to diminish hallucinations in psychotic individuals.

    More
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