参考文献
[1] Cho et al (1998) Discovery of a novel, potent, and orally active nonpeptide antagonist of the human luteinizing hormone-releasing hormone (LHRH) receptor. J.Med.Chem. 41 4190. PMID: 9784092.
[2] Sasaki et al (2003) Discovery of a thieno[2,3-d]pyrimidine-2,4-dione bearing a p-methoxyureidophenyl moiety at the 6-position: a highly potent and orally bioavailable non-peptide antagonist for the human luteinizing hormone-releasing hormone receptor. J.Med.Chem. 46 113. PMID: 12502365.
[3] Imada et al (2006) Design, synthesis, and structure-activity relationships of thieno[2,3-b]pyridin-4-one derivatives as a novel class of potent, orally active, non-peptide luteinizing hormone-releasing hormone receptor antagonists. J.Med.Chem. 49 3809. PMID: 16789738.
分子式
C37H37F2N3O4S |
分子量
657.77 |
CAS号
199119-18-1 |
储存方式
﹣20 ℃长期储存。冰袋运输 |
溶剂（常温）
|
DMSO
50 mM |
Water
|
Ethanol
|
体内溶解度
