参考文献
[1] Emonds-Alt et al (1993) In vitro and in vivo biological activities of SR140333, a novel non-peptide tachykinin NK1 receptor antagonist. Eur.J.Pharmacol. 250 403. PMID: 7509286.
[2] Oury-Donat et al (1994) SR 140333, a novel, selective, and potent nonpeptide antagonist of the NK1 tachykinin receptor: characterization on the U373MG cell line. J.Neurochem. 62 1399. PMID: 7510780.
[3] Hall and Brain (1994) Inhibition by SR140333 of NK1 tachykinin receptor-evoked, nitric oxide-dependent vasodilation in the hamster cheek pouch microvasculature in vivo. Br.J.Pharmacol. 113 522. PMID: 7530573.
[4] Nieuwmeyer et al (2006) Ava[L-Pro9,N-MeLeu10] substance P(7-11) (GR 73632) and Sar9, Met(O2)11 increase distention-induced peristalsis through activation of neurokinin-1 receptors on smooth muscle and interstitial cells of Cajal. J.Pharmacol.Exp.Ther. 317 439. PMID: 16330493.
分子式
C37H45Cl3N2O2 |
分子量
656.12 |
CAS号
153050-21-6 |
储存方式
﹣20 ℃长期储存。冰袋运输 |
溶剂（常温）
|
DMSO
100 mM |
Water
|
Ethanol
100 mM |
体内溶解度
