参考文献
[1] Williams et al (1994) 1-(((7,7-dimethyl-2(S)-(2(S)-amino-4-(methylsulfonyl)butyramido)bicyclo[2.2.1]-heptan-1(S)-yl)methyl)sulfonyl)-4-(2-methylphenyl)piperazine (L-368,899): an orally bioavailable, non-peptide oxytocin antagonist with potential utility for managing preterm labor. J.Med.Chem. 37 565. PMID: 8126695.
[2] Mann et al (2003) Attenuation of PGE2α release in ewes infused with the oxytocin antagonist L-368,899. Domest.Anim.Endocrinol. 25 255. PMID: 14550509.
[3] Quattropani et al (2005) Discovery and development of a new class of potent, selective, orally active oxytocin receptor antagonist. J.Med.Chem. 48 7882. PMID: 16302826.
[4] Borthwick (2010) Oral oxytocin antagonists. J.Med.Chem. 53 6525. PMID: 20550119.
分子式
C26H42N4O5S2.HCl |
分子量
591.23 |
CAS号
160312-62-9 |
储存方式
﹣20 ℃长期储存。冰袋运输 |
溶剂（常温）
|
DMSO
100 mM |
Water
|
Ethanol
|
体内溶解度
