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Anagrelide HCl

盐酸阿那格雷,BL-4162A

Anagrelide(BL4162A)盐酸盐对血小板增多症有效。

目录号
EY1622
EY1622
EY1622
EY1622
纯度
99.14%
99.14%
99.14%
99.14%
规格
5 mg
10 mg
50 mg
100 mg
原价
280
465
1720
3200
售价
280
465
1720
3200
库存
现货
现货
现货
现货
订购
订购
订购
订购
订购
订购
  • 生物活性

    Anagrelide is a drug used for the treatment of essential thrombocytosis.

  • 体外研究

  • 体内研究

  • 激酶实验

  • 细胞实验

  • 动物实验

  • 不同实验动物依据体表面积的等效剂量转换表(数据来源于FDA指南)

    动物 A (mg/kg) = 动物 B (mg/kg)×动物 B的Km系数/动物 AKm系数


    例如,已知某工具药用于小鼠的剂量为88 mg/kg , 则用于大鼠的剂量换算方法:将88 mg/kg 乘以小鼠的Km系数(3),再除以大鼠的Km系数(6),得到该药物用于大鼠的等效剂量44 mg/kg。


  • 参考文献

    [1] Tefferi A, et al. Semin Thromb Hemost, 1997, 23(4), 379-383.

    分子式
    C10H8Cl3N3O
    分子量
    292.55
    CAS号
    58579-51-4
    储存方式
    ﹣20 ℃冷藏长期储存。冰袋运输
    溶剂(常温)
    DMSO
    15 mg/mL
    Water
    <1 mg/mL
    Ethanol
    <1 mg/mL

    体内溶解度

  • Clinical Trial Information ( data from http://clinicaltrials.gov )

    NCT Number Conditions Interventions Sponsor/Collaborators Phases Start Date Last Updated
    NCT02076815 Essential Thrombocythemia Drug: Anagrelide retard|Drug: Thromboreductin AOP Orphan Pharmaceuticals AG Phase 3 2014-02-01 2015-07-27
    NCT01352585 Essential Thrombocythaemia Drug: Anagrelide hydrochloride Shire 2011-07-01 2014-06-27
    NCT02125318 Thrombocytosis|Myeloproliferative Neoplasms Drug: Anagrelide CR Galena Biopharma, Inc. Phase 2 2014-05-01 2017-02-23
    NCT00648765 Healthy Drug: Anagrelide Hydrochloride Capsules 1 mg|Drug: Agrylin Capsules 1 mg Mylan Pharmaceuticals Phase 1 2003-01-01 2008-03-31
    NCT00648024 Healthy Drug: Anagrelide Hydrochloride Capsules 1 mg|Drug: Agrylin Capsules 1 mg Mylan Pharmaceuticals Phase 1 2003-01-01 2008-03-31
    NCT01230775 Essential Thrombocythaemia Drug: Anagrelide retard|Drug: Placebo AOP Orphan Pharmaceuticals AG Phase 3 2010-12-01 2016-05-25
    NCT01552928 Healthy Drug: Anagrelide 0.5 mg|Drug: Anagrelide 2.5 mg|Drug: Moxifloxacin|Drug: Placebo Shire Phase 1 2012-03-01 2014-03-12
    NCT00413634 Essential Thrombocythaemia Drug: anagrelide hydrochloride Shire Phase 2 2006-08-01 2014-06-06
    NCT01065038 Essential Thrombocythaemia Drug: Anagrelide|Drug: Hydroxyurea AOP Orphan Pharmaceuticals AG Phase 3 2002-09-01 2010-10-05
    NCT00202644 Thrombocythemia, Hemorrhagic Drug: Anagrelide|Drug: Hydroxyurea Shire Phase 4 2006-01-01 2016-02-18
    NCT01467661 Essential Thrombocythemia (ET) Drug: SPD422 (anagrelide hydrochloride) Shire Phase 3 2011-11-01 2016-06-22
    NCT00567502 Thrombocythemia, Essential Shire 2005-05-01 2015-10-15
    NCT01192347 Essential Thrombocythemia Shire 2010-09-01 2014-02-14
    NCT01214915 Thrombocythemia, Essential Drug: Anagrelide Hydrochloride Shire Phase 3 2010-11-01 2013-09-27
    NCT02962388 Essential Thrombocythemia Drug: Anagrelide|Drug: Ruxolitinib (JAKAVI庐)|Drug: IFN/ PegIFN French Innovative Leukemia Organisation|Novartis Pharmaceuticals Phase 2|Phase 3 2017-01-01 2017-01-16
    NCT02577926 Polycythemia Vera (PV)|Essential Thrombocythemia (ET) Drug: Ruxolitinib|Drug: BAT RWTH Aachen University|Novartis Phase 3 2015-10-01 2016-09-07
    NCT02038036 Polycythemia Vera Drug: Best Available Therapy|Drug: ruxolitinib Novartis Pharmaceuticals|Novartis Phase 3 2014-03-25 2017-03-07
    NCT01668173 Myeloproliferative Neoplasms Drug: AUY922 Memorial Sloan Kettering Cancer Center|Novartis Phase 2 2012-08-01 2016-04-11
    NCT02101268 Primary Myelofibrosis (PMF)|Post-polycythemia Vera (Post-PV)|Post-essential Thrombocythemia Myelofibrosis (Post-ET MF) Drug: Momelotinib|Drug: Best Available Therapy (BAT) Gilead Sciences Phase 3 2014-06-01 2017-02-13
    NCT02252159 Polycythemia Vera Incyte Corporation 2014-07-01 2017-02-28
    NCT01243944 Polycythemia Vera Drug: ruxolitinib tablets|Other: Best Available Therapy (BAT) Incyte Corporation|Novartis Pharmaceuticals Phase 3 2010-10-01 2016-09-21
    NCT00481052 Chronic Myeloid Leukemia Drug: Nilotinib Gruppo Italiano Malattie EMatologiche dell'Adulto Phase 2 2007-06-01 2016-10-24

    注:以上所有数据均来自公开文献,并不保证对所有实验均有效,数据仅供参考。

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