Anagrelide(BL4162A)盐酸盐对血小板增多症有效。
Anagrelide is a drug used for the treatment of essential thrombocytosis.
动物 A (mg/kg) = 动物 B (mg/kg)×动物 B的Km系数/动物 A的Km系数 | |
例如,已知某工具药用于小鼠的剂量为88 mg/kg , 则用于大鼠的剂量换算方法:将88 mg/kg 乘以小鼠的Km系数(3),再除以大鼠的Km系数(6),得到该药物用于大鼠的等效剂量44 mg/kg。
[1] Tefferi A, et al. Semin Thromb Hemost, 1997, 23(4), 379-383.
分子式 C10H8Cl3N3O |
分子量 292.55 |
CAS号 58579-51-4 |
储存方式 ﹣20 ℃冷藏长期储存。冰袋运输 |
溶剂(常温) |
DMSO 15 mg/mL |
Water <1 mg/mL |
Ethanol <1 mg/mL |
体内溶解度
NCT Number | Conditions | Interventions | Sponsor/Collaborators | Phases | Start Date | Last Updated |
NCT02076815 | Essential Thrombocythemia | Drug: Anagrelide retard|Drug: Thromboreductin | AOP Orphan Pharmaceuticals AG | Phase 3 | 2014-02-01 | 2015-07-27 |
NCT01352585 | Essential Thrombocythaemia | Drug: Anagrelide hydrochloride | Shire | 2011-07-01 | 2014-06-27 | |
NCT02125318 | Thrombocytosis|Myeloproliferative Neoplasms | Drug: Anagrelide CR | Galena Biopharma, Inc. | Phase 2 | 2014-05-01 | 2017-02-23 |
NCT00648765 | Healthy | Drug: Anagrelide Hydrochloride Capsules 1 mg|Drug: Agrylin Capsules 1 mg | Mylan Pharmaceuticals | Phase 1 | 2003-01-01 | 2008-03-31 |
NCT00648024 | Healthy | Drug: Anagrelide Hydrochloride Capsules 1 mg|Drug: Agrylin Capsules 1 mg | Mylan Pharmaceuticals | Phase 1 | 2003-01-01 | 2008-03-31 |
NCT01230775 | Essential Thrombocythaemia | Drug: Anagrelide retard|Drug: Placebo | AOP Orphan Pharmaceuticals AG | Phase 3 | 2010-12-01 | 2016-05-25 |
NCT01552928 | Healthy | Drug: Anagrelide 0.5 mg|Drug: Anagrelide 2.5 mg|Drug: Moxifloxacin|Drug: Placebo | Shire | Phase 1 | 2012-03-01 | 2014-03-12 |
NCT00413634 | Essential Thrombocythaemia | Drug: anagrelide hydrochloride | Shire | Phase 2 | 2006-08-01 | 2014-06-06 |
NCT01065038 | Essential Thrombocythaemia | Drug: Anagrelide|Drug: Hydroxyurea | AOP Orphan Pharmaceuticals AG | Phase 3 | 2002-09-01 | 2010-10-05 |
NCT00202644 | Thrombocythemia, Hemorrhagic | Drug: Anagrelide|Drug: Hydroxyurea | Shire | Phase 4 | 2006-01-01 | 2016-02-18 |
NCT01467661 | Essential Thrombocythemia (ET) | Drug: SPD422 (anagrelide hydrochloride) | Shire | Phase 3 | 2011-11-01 | 2016-06-22 |
NCT00567502 | Thrombocythemia, Essential | Shire | 2005-05-01 | 2015-10-15 | ||
NCT01192347 | Essential Thrombocythemia | Shire | 2010-09-01 | 2014-02-14 | ||
NCT01214915 | Thrombocythemia, Essential | Drug: Anagrelide Hydrochloride | Shire | Phase 3 | 2010-11-01 | 2013-09-27 |
NCT02962388 | Essential Thrombocythemia | Drug: Anagrelide|Drug: Ruxolitinib (JAKAVI庐)|Drug: IFN/ PegIFN | French Innovative Leukemia Organisation|Novartis Pharmaceuticals | Phase 2|Phase 3 | 2017-01-01 | 2017-01-16 |
NCT02577926 | Polycythemia Vera (PV)|Essential Thrombocythemia (ET) | Drug: Ruxolitinib|Drug: BAT | RWTH Aachen University|Novartis | Phase 3 | 2015-10-01 | 2016-09-07 |
NCT02038036 | Polycythemia Vera | Drug: Best Available Therapy|Drug: ruxolitinib | Novartis Pharmaceuticals|Novartis | Phase 3 | 2014-03-25 | 2017-03-07 |
NCT01668173 | Myeloproliferative Neoplasms | Drug: AUY922 | Memorial Sloan Kettering Cancer Center|Novartis | Phase 2 | 2012-08-01 | 2016-04-11 |
NCT02101268 | Primary Myelofibrosis (PMF)|Post-polycythemia Vera (Post-PV)|Post-essential Thrombocythemia Myelofibrosis (Post-ET MF) | Drug: Momelotinib|Drug: Best Available Therapy (BAT) | Gilead Sciences | Phase 3 | 2014-06-01 | 2017-02-13 |
NCT02252159 | Polycythemia Vera | Incyte Corporation | 2014-07-01 | 2017-02-28 | ||
NCT01243944 | Polycythemia Vera | Drug: ruxolitinib tablets|Other: Best Available Therapy (BAT) | Incyte Corporation|Novartis Pharmaceuticals | Phase 3 | 2010-10-01 | 2016-09-21 |
NCT00481052 | Chronic Myeloid Leukemia | Drug: Nilotinib | Gruppo Italiano Malattie EMatologiche dell'Adulto | Phase 2 | 2007-06-01 | 2016-10-24 |
注:以上所有数据均来自公开文献,并不保证对所有实验均有效,数据仅供参考。
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