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Tetracycline HCl

盐酸四环素,NCI-c55561,Sumycin,NCI-c 55561,NCI-c-55561,

Tetracycline hydrochloride 是广谱聚酮类抗生素。

目录号
EY1537
EY1537
EY1537
纯度
99.15%
99.15%
99.15%
规格
500 mg
1 g
5 g
原价
315
398
780
售价
315
398
780
库存
现货
现货
现货
订购
订购
订购
订购
订购
订购
  • 生物活性

    Tetracycline HCl is a hydrochloride salt of tetracycline that is a broad-spectrum polyketide antibiotic.

  • 体外研究

  • 体内研究

  • 激酶实验

  • 细胞实验

  • 动物实验

  • 不同实验动物依据体表面积的等效剂量转换表(数据来源于FDA指南)

    动物 A (mg/kg) = 动物 B (mg/kg)×动物 B的Km系数/动物 AKm系数


    例如,已知某工具药用于小鼠的剂量为88 mg/kg , 则用于大鼠的剂量换算方法:将88 mg/kg 乘以小鼠的Km系数(3),再除以大鼠的Km系数(6),得到该药物用于大鼠的等效剂量44 mg/kg。


  • 参考文献

    [1] E Kheadr et. Al. Antimicrobial Agents and Chemotherapy, 51(1), 169-174 (2007).
    [2] Hyekyung P Cho et. Al. ACS Chemical Neuroscience, 5(7), 597-610 (2014).
    [3] Yuqin Qiao et. Al. Biomaterials, 35(25), 6882-6897 (2014).

    分子式
    C22H25ClN2O8
    分子量
    480.9
    CAS号
    64-75-5
    储存方式
    ﹣20 ℃冷藏长期储存。冰袋运输
    溶剂(常温)
    DMSO
    100 mg/mL
    Water
    100 mg/mL
    Ethanol
    <1 mg/mL

    体内溶解度

  • Clinical Trial Information ( data from http://clinicaltrials.gov )

    NCT Number Conditions Interventions Sponsor/Collaborators Phases Start Date Last Updated
    NCT01880515 Skin Rash|Lung Cancer Drug: Tetracycline Instituto Nacional de Cancerologia de Mexico Phase 2 2010-12-01 2014-01-15
    NCT01763437 Chalazia|Chalazion Drug: Tetracycline The Cleveland Clinic Early Phase 1 2014-03-01 2017-01-10
    NCT02057926 Ridge Preservation Technique Drug: The effect of tetracycline in degradation and permeability of collagen membranes. Universitat Internacional de Catalunya Phase 2 2009-11-01 2014-02-05
    NCT02259543 Gingival Recession Other: Root conditioning with citric acid+tetracycline solution University of Sao Paulo|Fundao de Amparo Pesquisa do Estado de So Paulo 2011-08-01 2014-10-05
    NCT00091247 Unspecified Adult Solid Tumor, Protocol Specific Drug: tetracycline hydrochloride|Other: placebo Alliance for Clinical Trials in Oncology|National Cancer Institute (NCI) 2004-12-01 2017-03-14
    NCT00336154 Epidermolysis Bullosa Drug: tetracyclin Rambam Health Care Campus Phase 4 2006-06-12
    NCT00355459 Dry Eye Syndrome Drug: Tetracycline: Doxycycline analog University of Texas Southwestern Medical Center 2005-08-01 2011-03-21
    NCT01293643 Vaginosis, Bacterial|Candidiasis, Vulvovaginal Drug: 100 mg clindamycin /800 mg ketoconazole vaginal ovule|Drug: 100 mg tetracycline hydrochloride /50 mg amphotericin B cream Merck Sharp & Dohme Corp. Phase 3 2010-05-01 2015-08-07
    NCT02175927 Helicobacter Pylori Treatment Failure Drug: Lansoprazole|Drug: Bismuth Potassium Citrate|Drug: Metronidazole|Drug: Amoxicillin|Drug: Tetracycline Shanghai Jiao Tong University School of Medicine Phase 4 2014-07-01 2016-02-29
    NCT00469261 Myocardial Infarction|Left Ventricular Remodeling Drug: Doxycycline|Drug: Current medical therapy for AMI Careggi Hospital Phase 2 2007-05-01 2012-09-24
    NCT00669955 Helicobacter Infections Drug: Omeprazole, amoxicillin, clarithromycin|Drug: Pylera (Bismuth subcitrate potassium, metronidazole, tetracycline) given in combination with omeprazole Forest Laboratories Phase 3 2008-06-01 2017-02-08
    NCT00889356 Candidiasis|Bacterial Vaginosis Drug: Clindamycin 100mg and Ketoconazole 400mg|Drug: Tetracycline 100mg and Amphotericin B 50mg Zodiac Produtos Farmaceuticos S.A. Phase 3 2009-09-01 2009-04-27
    NCT02576652 Osteoporosis Other: Tetracycline/Demeclocycline Amgen Phase 4 2015-12-01 2016-12-07
    NCT02978157 Helicobacter Pylori Infection Drug: esomeprazole+amox+levo|Drug: esomeprazole+bismuth+tetra+levo Kaohsiung Veterans General Hospital.|Kaohsiung Medical University Chung-Ho Memorial Hospital 2015-02-01 2016-11-29
    NCT01573975 Helicobacter Pylori Infection Drug: 5RA-5RCM|Drug: 5RA-5RCT|Drug: 10RCA Buddhist Tzu Chi General Hospital Phase 4 2009-01-01 2012-04-09
    NCT00243893 Aneurysms|Arteriovenous Malformations Drug: minocycline|Drug: doxycycline University of California, San Francisco|National Institute of Neurological Disorders and Stroke (NINDS) Phase 1 2004-07-01 2013-10-08
    NCT00347776 Trichiasis Drug: azithromycin|Drug: topical tetracycline Johns Hopkins University|National Eye Institute (NEI)|Project ORBIS Phase 4 2001-08-01 2013-04-03
    NCT01010295 Non-Hodgkin Lymphoma Drug: doxycycline (tetracycline) International Extranodal Lymphoma Study Group (IELSG) Phase 2 2006-09-01 2013-11-22
    NCT01335334 H. Pylori Infection Drug: bismuth subcitrate potassium, metronidazole,tetracycline hydrochloride and omeprazole The University of Texas Health Science Center, Houston Phase 4 2011-03-01 2011-04-13
    NCT00591162 Burn Drug: Tetracycline|Radiation: Duel Energy X-Ray Absorptiometry (DEXA)|Procedure: Bone Biopsy The University of Texas Medical Branch, Galveston Phase 2|Phase 3 1992-10-01 2014-06-05

    注:以上所有数据均来自公开文献,并不保证对所有实验均有效,数据仅供参考。

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