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Solifenacin succinate

琥珀酸索非那新,YM905,YM-905,YM 905

Solifenacin Succinate (琥珀酸索利那新; YM905; Vesicare) 是毒蕈碱受体拮抗剂。

目录号
EY1399
EY1399
EY1399
纯度
99.61%
99.61%
99.61%
规格
10 mg
50 mg
100 mg
原价
290
580
1020
售价
290
580
1020
库存
现货
现货
现货
订购
订购
订购
订购
订购
订购
  • 生物活性

    Solifenacin succinate is a urinary antispasmodic of the antimuscarinic class.

  • 体外研究

  • 体内研究

  • 激酶实验

  • 细胞实验

  • 动物实验

  • 不同实验动物依据体表面积的等效剂量转换表(数据来源于FDA指南)

    动物 A (mg/kg) = 动物 B (mg/kg)×动物 B的Km系数/动物 AKm系数


    例如,已知某工具药用于小鼠的剂量为88 mg/kg , 则用于大鼠的剂量换算方法:将88 mg/kg 乘以小鼠的Km系数(3),再除以大鼠的Km系数(6),得到该药物用于大鼠的等效剂量44 mg/kg。


  • 参考文献

    [1] Ikeda K, et al. Naunyn Schmiedebergs Arch Pharmacol, 2002, 366(2), 97-103.

    分子式
    C27H32N2O6
    分子量
    480.55
    CAS号
    242478-38-2
    储存方式
    ﹣20 ℃冷藏长期储存。冰袋运输
    溶剂(常温)
    DMSO
    3 mg/mL
    Water
    96 mg/mL
    Ethanol
    5 mg/mL

    体内溶解度

  • Clinical Trial Information ( data from http://clinicaltrials.gov )

    NCT Number Conditions Interventions Sponsor/Collaborators Phases Start Date Last Updated
    NCT01015040 Bioavailability of Solifenacin Succinate|Pharmacokinetics of Solifenacin Succinate|Healthy Volunteers Drug: solifenacin succinate suspension|Drug: solifenacin succinate tablet Astellas Pharma Inc Phase 1 2009-09-01 2009-12-04
    NCT01371994 Urinary Incontinence Drug: solifenacin succinate|Drug: Placebo Astellas Pharma Inc Phase 4 2011-08-01 2014-10-06
    NCT01539707 Overactive Bladder|Neurogenic Detrusor Overactivity Drug: Solifenacin succinate Astellas Pharma Inc Phase 1 2012-03-01 2012-10-29
    NCT00454740 Urinary Bladder, Overactive Drug: solifenacin succinate Astellas Pharma Inc Phase 3 2004-06-01 2014-09-17
    NCT00463541 Urinary Bladder, Overactive Drug: solifenacin succinate Astellas Pharma Inc Phase 3 2004-06-01 2014-09-17
    NCT00773552 Urinary Urge|Urge Incontinence|Overactive Bladder Drug: solifenacin succinate|Drug: placebo Stamford Hospital Phase 4 2008-11-01 2016-12-05
    NCT00985387 Urinary Bladder, Overactive|Overactive Bladder Drug: Solifenacin Astellas Pharma Inc|Astellas Pharma Korea, Inc. 2009-08-01 2011-10-11
    NCT01981954 Neurogenic Detrusor Overactivity|Pediatric Drug: Solifenacin succinate Astellas Pharma Europe B.V.|Astellas Pharma Inc Phase 3 2013-09-01 2016-06-02
    NCT00507455 Lower Urinary Tract Symptoms|Bladder Outlet Obstruction Drug: solifenacin succinate|Drug: tamsulosin hydrochloride|Drug: Placebo to solifenacin|Drug: Placebo to tamsulosin Astellas Pharma Inc Phase 2 2007-06-01 2014-07-14
    NCT01565707 Urinary Bladder, Overactive Drug: Solifenacin Succinate Suspension|Drug: Placebo|Behavioral: Urotherapy Astellas Pharma Europe B.V.|Astellas Pharma Inc Phase 3 2012-06-01 2016-12-05
    NCT01777217 Over-Active Bladder Drug: Solifenacin succinate|Drug: Placebo Advanced Research Network|Astellas Pharma US, Inc. Phase 4 2013-02-01 2015-01-08
    NCT01833663 Overactive Bladder|Postmenopausal Disorder|Urination Disorders Drug: Solifenacin Succinate Tablets|Drug: Estrogen Peking Union Medical College Hospital|Astellas Pharma China, Inc.|Beijing CAT Science Co., Ltd. Phase 4 2011-10-01 2014-03-19
    NCT01655069 Urinary Bladder, Overactive Drug: Solifenacin succinate Astellas Pharma Europe B.V.|Astellas Pharma Inc Phase 3 2012-10-01 2015-07-23
    NCT01406158 Pharmacokinetics of Solifenacin Succinate|Healthy Volunteers Drug: Solifenacin Succinate Formulation A|Drug: Solifenacin Succinate Formulation B|Drug: Solifenacin Succinate Astellas Pharma Inc Phase 1 2011-05-01 2011-08-23
    NCT01595152 Urinary Bladder, Overactive Drug: solifenacin succinate|Drug: fesoterodine Rambam Health Care Campus 2012-05-01 2012-05-14
    NCT00454896 Urinary Bladder, Overactive Drug: VESIcare|Drug: placebo Astellas Pharma Inc Phase 3 2004-05-01 2014-09-17
    NCT01565694 Neurogenic Detrusor Overactivity Drug: Solifenacin succinate Astellas Pharma Europe B.V.|Astellas Pharma Inc Phase 3 2012-09-01 2016-07-24
    NCT01093534 Detrusor Overactivity|Overactive Bladder Drug: Placebo|Drug: solifenacin Astellas Pharma Inc Phase 4 2010-01-01 2017-02-15
    NCT00337558 Overactive Bladder|Urinary Incontinence|Urge Incontinence Drug: Solifenacin succinate|Behavioral: Simplified bladder training Astellas Pharma Inc|Astellas Pharma Europe B.V. Phase 4 2006-05-01 2014-09-17
    NCT02010944 Phase 1|Bioavailability|Healthy Subjects Drug: solifenacin succinate|Drug: mirabegron|Drug: mirabegron/solifenacin succinate Astellas Pharma Europe B.V.|Astellas Pharma Inc Phase 1 2012-09-01 2013-12-10
    NCT00884104 Overactive Bladder Drug: Solifenacin KYU-SUNG LEE|Astellas Pharma Korea, Inc.|Samsung Medical Center Phase 4 2009-03-01 2016-01-06

    注:以上所有数据均来自公开文献,并不保证对所有实验均有效,数据仅供参考。

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