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FPH2

BRD-9424,BRD 9424,BRD9424,FPH-2,FPH 2,

FPH2 (BRD-9424) 是一种小分子,可促进iPS衍生肝细胞的分化。

目录号
EY1335
EY1335
EY1335
EY1335
纯度
99.48%
99.48%
99.48%
99.48%
规格
5 mg
10 mg
25 mg
50 mg
原价
450
790
1600
2900
售价
450
790
1600
2900
库存
现货
现货
现货
现货
订购
订购
订购
订购
订购
订购
  • 生物活性

    FPH2 (BRD-9424) is a small molecule, which promotes differentiation of iPS-derived hepatocytes.

  • 体外研究

  • 体内研究

  • 激酶实验

  • 细胞实验

  • 动物实验

  • 不同实验动物依据体表面积的等效剂量转换表(数据来源于FDA指南)

    动物 A (mg/kg) = 动物 B (mg/kg)×动物 B的Km系数/动物 AKm系数


    例如,已知某工具药用于小鼠的剂量为88 mg/kg , 则用于大鼠的剂量换算方法:将88 mg/kg 乘以小鼠的Km系数(3),再除以大鼠的Km系数(6),得到该药物用于大鼠的等效剂量44 mg/kg。


  • 参考文献

    [1] Shan J, et al. Nat Chem Biol. 2013, 9(8), 514-520.

    分子式
    分子量
    CAS号
    957485-64-2
    储存方式
    ﹣20 ℃冷藏长期储存。冰袋运输
    溶剂(常温)
    DMSO
    70 mg/mL
    Water
    <1 mg/mL
    Ethanol
    <1 mg/mL

    体内溶解度

  • Clinical Trial Information ( data from http://clinicaltrials.gov )

    NCT Number Conditions Interventions Sponsor/Collaborators Phases Start Date Last Updated
    NCT00001398 Aplastic Anemia|Pancytopenia Drug: Recombinant Methionyl Human Stem Cell Factor (r-metHuSCF) National Heart, Lung, and Blood Institute (NHLBI)|National Institutes of Health Clinical Center (CC) Phase 1 1993-10-01 2008-03-03
    NCT00005783 Hemoglobin SC Disease|Sickle Cell Anemia Drug: Recombinant-methionyl human stem cell factor National Institute of Diabetes and Digestive and Kidney Diseases (NIDDK)|National Institutes of Health Clinical Center (CC) Phase 1 2000-03-01 2008-03-03
    NCT00058045 Lymphoma Biological: aldesleukin|Biological: recombinant human stem cell factor Roswell Park Cancer Institute|National Cancer Institute (NCI) Phase 1 2002-08-01 2013-01-30
    NCT00434239 Myelodysplasia Drug: Lenalidomide + Ancestim Peter MacCallum Cancer Centre, Australia|Celgene Corporation Early Phase 1 2007-02-01 2013-01-08
    NCT00005993 Breast Cancer|Lymphoma Drug: aldesleukin|Drug: filgrastim|Drug: recombinant human stem cell factor|Procedure: peripheral blood stem cell transplantation Masonic Cancer Center, University of Minnesota|National Cancer Institute (NCI) Phase 1 1999-05-01 2012-10-09
    NCT01016795 Malignant Lymphoma Drug: r-metHuSCF and Filgrastim|Drug: r-metHuSCF and Filgrastim|Drug: Chemotherapy plus Filgrastim Aalborg Universitetshospital|Herlev Hospital|Rigshospitalet, Denmark|Helsinki University Central Hospital|Turku University Hospital|University Hospital, Linkoeping|Ume University|Oslo University Hospital|Nordic Lymphoma Group|Amgen Phase 2 1999-01-01 2015-06-24
    NCT00001750 Multiple Myeloma Drug: Stemgen National Heart, Lung, and Blood Institute (NHLBI)|National Institutes of Health Clinical Center (CC) Phase 2 1998-09-01 2008-03-03
    NCT02553304 Chronic Lymphocytic Leukemia (CLL) National Health Research Institutes, Taiwan 2015-09-01 2016-01-13
    NCT00154466 Myocardial Infarction Behavioral: cardiac rehabilitation National Taiwan University Hospital 2004-07-01 2014-05-25
    NCT00001356 Mastocytosis National Institute of Allergy and Infectious Diseases (NIAID)|National Institutes of Health Clinical Center (CC) 1993-05-01 2008-03-03
    NCT00216112 Ovarian Cancer Drug: Imatinib Mesylate|Drug: Docetaxel Daniela Matei, MD|Novartis Pharmaceuticals|Sanofi|Walther Cancer Institute|Hoosier Cancer Research Network Phase 2 2003-12-01 2016-02-17
    NCT02461849 Advanced, Refractory Cancer Drug: Imatinib Samsung Medical Center Phase 2 2014-04-04 2017-02-15
    NCT01440959 Gastrointestinal Stromal Tumors Drug: dovitinib Asan Medical Center Phase 2 2011-09-01 2014-01-13
    NCT01563822 Intra-cytoplasmic Sperm Injection Outcome Biological: Follicular fluid Nawara Mohamed Hashish|Kasr El Aini Hospital Phase 1 2011-12-01 2012-10-06
    NCT00731744 Normal Full-Term Deliveries Procedure: Normal full-term deliveries National Taiwan University Hospital 2007-01-01 2008-08-08
    NCT01222143 Acute Myeloid Leukemia Drug: NOVE-HiDAC|Drug: Nilotinib University Health Network, Toronto|Novartis Pharmaceuticals Phase 1|Phase 2 2010-10-01 2015-06-19
    NCT02145897 Critical Limb Ischemia Biological: Autologous Stromal Vascular Fraction (SVF)|Biological: Autologous Adipose Derieved MSCs|Other: Control Kasiak Research Pvt. Ltd. Phase 1|Phase 2 2014-08-01 2014-05-20
    NCT01172548 Gastrointestinal Stromal Tumors Drug: imatinib mesylate Novartis Pharmaceuticals|Novartis Phase 2 2008-08-01 2017-02-24
    NCT01624701 Acute Leukemia|Chronic Leukemia|Myelodysplastic Syndrome|Lymphoma|Myeloma Other: Ex vivo expanded cord blood cells Singapore General Hospital|Whitehead Institute for Biomedical Research|Blood Services Group, Health Sciences Authority of Singapore Phase 1|Phase 2 2012-03-01 2015-11-26
    NCT02148367 Traumatic Brain Injury Drug: Erythropoietin Uniformed Services University of the Health Sciences|National Institutes of Health (NIH) Phase 2 2014-09-01 2015-12-30
    NCT00003957 Lymphoma Biological: filgrastim|Biological: recombinant human stem cell factor|Drug: cyclophosphamide|Drug: cytarabine|Drug: etoposide|Drug: melphalan|Drug: mitoxantrone hydrochloride|Drug: paclitaxel|Procedure: peripheral blood stem cell transplantation Fox Chase Cancer Center|National Cancer Institute (NCI) Phase 2 1998-12-01 2013-04-16
    NCT03033953 Healthy|Young|Elderly Dietary Supplement: Native whey|Dietary Supplement: Milk|Other: Strength training Norwegian School of Sport Sciences|Tine|The Research Council of Norway 2014-08-01 2017-01-24
    NCT00001760 Atopic Dermatitis|Healthy|Mastocytosis National Institute of Allergy and Infectious Diseases (NIAID)|National Institutes of Health Clinical Center (CC) 1998-01-01 2007-12-12
    NCT00457743 Gastrointestinal Stromal Tumors Drug: Sunitinib malate (SU011248) Pfizer Phase 1|Phase 2 2005-01-01 2009-10-02
    NCT00569946 Carcinoma, Renal Cell Drug: AG-013736 Pfizer Phase 2 2007-12-01 2014-07-16

    注:以上所有数据均来自公开文献,并不保证对所有实验均有效,数据仅供参考。

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