Amlodipine besylate是长效钙离子通道抑制剂。
Amlodipine Besylate is a long-acting calcium channel blocker, used to lower blood pressure and prevent chest pain.
动物 A (mg/kg) = 动物 B (mg/kg)×动物 B的Km系数/动物 A的Km系数 | |
例如,已知某工具药用于小鼠的剂量为88 mg/kg , 则用于大鼠的剂量换算方法:将88 mg/kg 乘以小鼠的Km系数(3),再除以大鼠的Km系数(6),得到该药物用于大鼠的等效剂量44 mg/kg。
[1] Lee YJ, et al. J Neurochem, 2011, 119(6), 1262-1270.
分子式 C26H31ClN2O8S |
分子量 567.05 |
CAS号 111470-99-6 |
储存方式 ﹣20 ℃冷藏长期储存。冰袋运输 |
溶剂(常温) |
DMSO ≥20 mg/mL |
Water <1 mg/mL |
Ethanol ≥14 mg/mL |
体内溶解度
NCT Number | Conditions | Interventions | Sponsor/Collaborators | Phases | Start Date | Last Updated |
NCT01155908 | Healthy | Drug: Amlodipine Besylate / Benazepril Hydrochloride | Dr. Reddy's Laboratories Limited | Phase 1 | 2005-04-01 | 2010-07-01 |
NCT02353806 | Chronic Hypertension in Pregnancy | Drug: Amlodipine besylate | University of Texas Southwestern Medical Center|National Center for Advancing Translational Science (NCATS) | Phase 4 | 2015-01-01 | 2016-05-10 |
NCT01155895 | Healthy | Drug: Amlodipine Besylate / Benazepril Hydrochloride | Dr. Reddy's Laboratories Limited | Phase 1 | 2004-03-01 | 2010-07-01 |
NCT01131936 | Healthy | Drug: Amlodipine | Dr. Reddy's Laboratories Limited | Phase 1 | 2002-08-01 | 2010-06-11 |
NCT01131923 | Healthy | Drug: Amlodipine | Dr. Reddy's Laboratories Limited | Phase 1 | 2002-10-01 | 2010-06-11 |
NCT02940548 | Hypertension | Drug: Nifedipine GITS|Drug: Amlodipine besylate | Jing Liu|Bayer|Peking University People's Hospital | Phase 4 | 2016-12-01 | 2016-12-13 |
NCT02707913 | Healthy | Drug: BF-Amlodipine Tablet 10mg|Drug: Norvasc Tablet 10mg | Bright Future Pharmaceuticals Factory O/B Bright Future Pharmaceutical Laboratories Limited|Chinese University of Hong Kong | Phase 1 | 2016-03-01 | 2016-09-05 |
NCT02064556 | Hypertension | Drug: Amlodipine 10mg|Drug: Amlodipine 10mg/Candesartan 32mg | Chong Kun Dang Pharmaceutical | Phase 1 | 2014-05-01 | 2014-08-13 |
NCT01845272 | Healthy | Drug: candesartan cilexetil 32mg, amlodipine 10mg|Drug: candesartan cilexetil 32mg, amlodipine 10mg | CJ HealthCare Corporation | Phase 1 | 2013-04-01 | 2013-04-30 |
NCT00870142 | Healthy | Drug: AMLODIPINE (as BESILATE) TABLETS 10 mg , single dose|Drug: Norvasc庐 10 mg Tablets | Actavis Inc. | Phase 1 | 2005-04-01 | 2010-08-13 |
NCT00870571 | Healthy | Drug: AMLODIPINE (as BESILATE) TABLETS 10 mg , single dose|Drug: NorvasC庐 10 mg Tablets | Actavis Inc. | Phase 1 | 2005-04-01 | 2010-08-13 |
NCT01505998 | Fed | Drug: Amlodipine Besylate/Benazepril HCl | Dr. Reddy's Laboratories Limited | Phase 1 | 2007-03-01 | 2012-01-06 |
NCT01506011 | Fasting | Drug: Amlodipine Besylate/Benazepril HCl | Dr. Reddy's Laboratories Limited | Phase 1 | 2007-03-01 | 2012-01-05 |
NCT02974439 | Bioequivalence | Drug: LANDI-Amlodipine Besylate Tablet 5mg|Drug: Norvasc Tablets 5mg | Shanghai Haini Pharmaceutical Co., Ltd. | Phase 1 | 2016-12-01 | 2017-02-13 |
NCT02292069 | Healthy | Drug: Amlodipine besylate/Atorvastatin calcium | Dr. Reddy's Laboratories Limited | Phase 1 | 2011-09-01 | 2014-11-12 |
NCT02295046 | Healthy | Drug: Amlodipine besylate/Atorvastatin calcium | Dr. Reddy's Laboratories Limited | Phase 1 | 2011-10-01 | 2014-11-17 |
NCT01252563 | Hypertension | Drug: Amlodipine | Pfizer | Phase 4 | 2010-12-01 | 2014-01-09 |
NCT00446524 | Hypertension | Drug: Valsartan + Amlodipine besilate | Novartis | Phase 3 | 2007-02-01 | 2012-05-06 |
注:以上所有数据均来自公开文献,并不保证对所有实验均有效,数据仅供参考。
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