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Amlodipine Besylate

苯磺酸氨氯地平

Amlodipine besylate是长效钙离子通道抑制剂。

目录号
EY1334
EY1334
EY1334
纯度
99.47%
99.47%
99.47%
规格
500 mg
1 g
5 g
原价
299
490
1060
售价
299
490
1060
库存
现货
现货
现货
订购
订购
订购
订购
订购
订购
  • 生物活性

    Amlodipine Besylate is a long-acting calcium channel blocker, used to lower blood pressure and prevent chest pain.

  • 体外研究

  • 体内研究

  • 激酶实验

  • 细胞实验

  • 动物实验

  • 不同实验动物依据体表面积的等效剂量转换表(数据来源于FDA指南)

    动物 A (mg/kg) = 动物 B (mg/kg)×动物 B的Km系数/动物 AKm系数


    例如,已知某工具药用于小鼠的剂量为88 mg/kg , 则用于大鼠的剂量换算方法:将88 mg/kg 乘以小鼠的Km系数(3),再除以大鼠的Km系数(6),得到该药物用于大鼠的等效剂量44 mg/kg。


  • 参考文献

    [1] Lee YJ, et al. J Neurochem, 2011, 119(6), 1262-1270.

    分子式
    C26H31ClN2O8S
    分子量
    567.05
    CAS号
    111470-99-6
    储存方式
    ﹣20 ℃冷藏长期储存。冰袋运输
    溶剂(常温)
    DMSO
    ≥20 mg/mL
    Water
    <1 mg/mL
    Ethanol
    ≥14 mg/mL

    体内溶解度

  • Clinical Trial Information ( data from http://clinicaltrials.gov )

    NCT Number Conditions Interventions Sponsor/Collaborators Phases Start Date Last Updated
    NCT01155908 Healthy Drug: Amlodipine Besylate / Benazepril Hydrochloride Dr. Reddy's Laboratories Limited Phase 1 2005-04-01 2010-07-01
    NCT02353806 Chronic Hypertension in Pregnancy Drug: Amlodipine besylate University of Texas Southwestern Medical Center|National Center for Advancing Translational Science (NCATS) Phase 4 2015-01-01 2016-05-10
    NCT01155895 Healthy Drug: Amlodipine Besylate / Benazepril Hydrochloride Dr. Reddy's Laboratories Limited Phase 1 2004-03-01 2010-07-01
    NCT01131936 Healthy Drug: Amlodipine Dr. Reddy's Laboratories Limited Phase 1 2002-08-01 2010-06-11
    NCT01131923 Healthy Drug: Amlodipine Dr. Reddy's Laboratories Limited Phase 1 2002-10-01 2010-06-11
    NCT02940548 Hypertension Drug: Nifedipine GITS|Drug: Amlodipine besylate Jing Liu|Bayer|Peking University People's Hospital Phase 4 2016-12-01 2016-12-13
    NCT02707913 Healthy Drug: BF-Amlodipine Tablet 10mg|Drug: Norvasc Tablet 10mg Bright Future Pharmaceuticals Factory O/B Bright Future Pharmaceutical Laboratories Limited|Chinese University of Hong Kong Phase 1 2016-03-01 2016-09-05
    NCT02064556 Hypertension Drug: Amlodipine 10mg|Drug: Amlodipine 10mg/Candesartan 32mg Chong Kun Dang Pharmaceutical Phase 1 2014-05-01 2014-08-13
    NCT01845272 Healthy Drug: candesartan cilexetil 32mg, amlodipine 10mg|Drug: candesartan cilexetil 32mg, amlodipine 10mg CJ HealthCare Corporation Phase 1 2013-04-01 2013-04-30
    NCT00870142 Healthy Drug: AMLODIPINE (as BESILATE) TABLETS 10 mg , single dose|Drug: Norvasc庐 10 mg Tablets Actavis Inc. Phase 1 2005-04-01 2010-08-13
    NCT00870571 Healthy Drug: AMLODIPINE (as BESILATE) TABLETS 10 mg , single dose|Drug: NorvasC庐 10 mg Tablets Actavis Inc. Phase 1 2005-04-01 2010-08-13
    NCT01505998 Fed Drug: Amlodipine Besylate/Benazepril HCl Dr. Reddy's Laboratories Limited Phase 1 2007-03-01 2012-01-06
    NCT01506011 Fasting Drug: Amlodipine Besylate/Benazepril HCl Dr. Reddy's Laboratories Limited Phase 1 2007-03-01 2012-01-05
    NCT02974439 Bioequivalence Drug: LANDI-Amlodipine Besylate Tablet 5mg|Drug: Norvasc Tablets 5mg Shanghai Haini Pharmaceutical Co., Ltd. Phase 1 2016-12-01 2017-02-13
    NCT02292069 Healthy Drug: Amlodipine besylate/Atorvastatin calcium Dr. Reddy's Laboratories Limited Phase 1 2011-09-01 2014-11-12
    NCT02295046 Healthy Drug: Amlodipine besylate/Atorvastatin calcium Dr. Reddy's Laboratories Limited Phase 1 2011-10-01 2014-11-17
    NCT01252563 Hypertension Drug: Amlodipine Pfizer Phase 4 2010-12-01 2014-01-09
    NCT00446524 Hypertension Drug: Valsartan + Amlodipine besilate Novartis Phase 3 2007-02-01 2012-05-06

    注:以上所有数据均来自公开文献,并不保证对所有实验均有效,数据仅供参考。

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