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Atropine

阿托品,Atropine sulfate hydrate

Atropine sulfate monohydrate是毒蕈碱乙酰胆碱受体拮抗剂。

目录号
EY1305
EY1305
纯度
99.61%
99.61%
规格
50 mg
100 mg
原价
270
485
售价
270
485
库存
现货
现货
订购
订购
订购
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  • 生物活性

    Atropine is a competitive antagonist for the muscarinic acetylcholine receptor, used to decrease the production of saliva and secretions of the airway prior to surgery.

  • 体外研究

  • 体内研究

  • 激酶实验

  • 细胞实验

  • 动物实验

  • 不同实验动物依据体表面积的等效剂量转换表(数据来源于FDA指南)

    动物 A (mg/kg) = 动物 B (mg/kg)×动物 B的Km系数/动物 AKm系数


    例如,已知某工具药用于小鼠的剂量为88 mg/kg , 则用于大鼠的剂量换算方法:将88 mg/kg 乘以小鼠的Km系数(3),再除以大鼠的Km系数(6),得到该药物用于大鼠的等效剂量44 mg/kg。


  • 参考文献

    [1] Schwahn HN, et al. Vis Neurosci,?000, 17(2), 165-176.

    分子式
    C34H50N2O11S
    分子量
    694.83
    CAS号
    5908-99-6
    储存方式
    ﹣20 ℃冷藏长期储存。冰袋运输
    溶剂(常温)
    DMSO
    200 mM
    Water
    200 mM
    Ethanol
    200 mM

    体内溶解度

  • Clinical Trial Information ( data from http://clinicaltrials.gov )

    NCT Number Conditions Interventions Sponsor/Collaborators Phases Start Date Last Updated
    NCT01819064 Bradycardia|Arrhythmias Drug: Atropine|Drug: Atropine State University of New York at Buffalo 2013-02-01 2013-08-01
    NCT02186132 Bradycardia|Neostigmine Adverse Reaction|Adverse Reaction to Belladonna or Atropine Drug: Atropine 0.6 mg|Drug: Atropine 1.2 mg Mahidol University Phase 4 2012-03-01 2014-07-07
    NCT00834470 Conscious Sedation Drug: Atropine Seoul National University Hospital Phase 4 2008-08-01 2012-08-03
    NCT02870478 Myopia Drug: Atropine University of California, Berkeley Phase 3 2016-07-01 2016-08-16
    NCT00947596 Organophosphorus Poisoning Drug: atropine sulfate|Drug: atropine sulfate MicroDose Defense Products L.L.C.|University of Pittsburgh|U.S. Army Space and Missile Defense Command Phase 1 2009-08-01 2010-08-10
    NCT02055378 Myopia Drug: Atropine|Device: auricular acupoint stimulation Taipei Tzu Chi Hospital, Buddhist Tzu Chi Medical Foundation 2011-01-01 2014-02-03
    NCT02130167 Myopia Progression Drug: Atropine Chang Gung Memorial Hospital 2012-08-01 2014-05-01
    NCT01595399 Bradycardia|Hypoxemia Drug: atropine|Drug: Placebo University of Manitoba Phase 4 2012-04-01 2013-09-23
    NCT00315302 Amblyopia Drug: Atropine|Device: Plano Lens Jaeb Center for Health Research|National Eye Institute (NEI) Phase 3 2005-02-01 2016-07-15
    NCT02704923 Ventilator-Associated Pneumonia Drug: Atropine|Drug: Placebo Universidade de Passo Fundo Phase 2 2015-02-01 2016-03-09
    NCT00623207 Chest Pain Drug: Atropine HaEmek Medical Center, Israel Phase 3 2007-12-01 2015-07-24
    NCT00944710 Amblyopia Drug: Atropine|Device: Plano lens|Drug: Atropine Jaeb Center for Health Research|National Eye Institute (NEI) Phase 3 2009-08-01 2016-07-07
    NCT00575523 Arrhythmia|Respiratory Arrest Drug: Atropine|Drug: Placebo Medical University of Vienna Phase 4 2003-10-01 2008-01-23
    NCT01464489 Intubation; Difficult Drug: Atropine|Drug: Normal saline Gachon University Gil Medical Center 2011-05-01 2011-11-01
    NCT02955927 Myopia Drug: 0.01% atropine eye drops|Device: ortho-k The Hong Kong Polytechnic University|The University of Hong Kong 2016-11-01 2016-11-03
    NCT00315328 Amblyopia Drug: Atropine|Device: Patching|Procedure: Near activities Jaeb Center for Health Research|National Eye Institute (NEI) Phase 3 2005-08-01 2016-05-19
    NCT02228473 Catheter Site Discomfort|Complications|Anesthesia|Urinary Bladder Neoplasms Drug: Glycopyrrolate|Drug: Atropine Seoul National University Hospital 2014-09-01 2014-10-27
    NCT01191398 Sialorrhea Drug: Atropine (0.01mg/kg)|Drug: Glycopyrrolate (0.01mg/kg)|Drug: Normal saline 0.9% Craig J. Huang|University of Texas Southwestern Medical Center 2010-06-01 2014-03-20
    NCT01871922 Anesthesia-induced Negative Hemodynamic Effects Drug: Placebo|Drug: Atropine University Medical Center Groningen 2012-10-01 2014-01-30
    NCT00921102 Cesarean Section|Anesthesia,Spinal|Postoperative Nausea and Vomiting Drug: Bupivacaine|Drug: Morphine|Drug: Isotonic saline solution|Drug: Atropine University of Parma Phase 4 2007-05-01 2009-06-15
    NCT00815048 Endotracheal Intubation Drug: Atropine/Remifentanil|Drug: Fentanyl/Atropine/Succinylcholine King Saud University|McMaster University Phase 4 2006-01-01 2008-12-26

    注:以上所有数据均来自公开文献,并不保证对所有实验均有效,数据仅供参考。

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