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Nystatin

制霉菌素,Fungicidin,Mycostatin

Nystatin是多烯类抗真菌抗生素,对酵母和支原体有效。

目录号
EY1240
EY1240
纯度
99.47%
99.47%
规格
250 mg
500 mg
原价
280
480
售价
280
480
库存
现货
现货
订购
订购
订购
订购
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  • 生物活性

    Nystatin, which belongs to the polyene group of antimycotics, is frequently used as a topical agent in the treatment of oro-pharyngeal candidosis.

  • 体外研究

  • 体内研究

  • 激酶实验

  • 细胞实验

  • 动物实验

  • 不同实验动物依据体表面积的等效剂量转换表(数据来源于FDA指南)

    动物 A (mg/kg) = 动物 B (mg/kg)×动物 B的Km系数/动物 AKm系数


    例如,已知某工具药用于小鼠的剂量为88 mg/kg , 则用于大鼠的剂量换算方法:将88 mg/kg 乘以小鼠的Km系数(3),再除以大鼠的Km系数(6),得到该药物用于大鼠的等效剂量44 mg/kg。


  • 参考文献

    [1] Brautaset, T., et al.: Chem. Biol., 7, 395 (2000), Brautaset, T., et al.: J. Biol. Chem., 278, 14913 (2003), Bruheim, P., et al.: Antimicrob. Agents Chemother., 48, 4120

    分子式
    C47H75NO17
    分子量
    926.09
    CAS号
    1400-61-9
    储存方式
    ﹣20 ℃冷藏长期储存。冰袋运输
    溶剂(常温)
    DMSO
    20 mg/mL
    Water
    <1 mg/mL
    Ethanol
    <1 mg/mL

    体内溶解度

  • Clinical Trial Information ( data from http://clinicaltrials.gov )

    NCT Number Conditions Interventions Sponsor/Collaborators Phases Start Date Last Updated
    NCT01198223 Denture Stomatitis Drug: garlic , nystatin Qazvin University Of Medical Sciences Phase 2 2010-07-01 2010-10-15
    NCT01495039 Fungal Prophylaxis|Candida Infection|Critical Illness|Surgery Drug: Nystatin Policlinico Hospital Phase 4 2008-11-01 2011-12-16
    NCT01427738 HIV-1 Infection Drug: Gentian Violet|Drug: Nystatin oral suspension AIDS Clinical Trials Group|National Institute of Allergy and Infectious Diseases (NIAID) Phase 3 2011-06-01 2015-02-12
    NCT00002097 HIV Infections Drug: Nystatin Argus Pharmaceuticals|NIH AIDS Clinical Trials Information Service Phase 1
    2005-06-23
    NCT00001998 HIV Infections Drug: Nystatin Argus Pharmaceuticals|NIH AIDS Clinical Trials Information Service
    2005-06-23
    NCT02186145 Bacterial Vaginosis|Fungal Vaginal Infections Drug: Association of metronidazole; nystatin and dexamethasone|Drug: Flagyl Marjan Industria e Comercio ltda Phase 3 2016-01-01 2015-04-08
    NCT00002057 Candidiasis, Oral|HIV Infections Drug: Nystatin Bristol-Myers Squibb
    2007-10-01
    NCT00002293 Candidiasis, Oral|HIV Infections Drug: Nystatin Bristol-Myers Squibb
    2007-10-01
    NCT02642900 Photochemotherapy Reaction Procedure: Photodynamic Therapy|Drug: Nystatin 100.000 units University of Sao Paulo Phase 4 2009-07-01 2015-12-25
    NCT00002313 HIV Infections Drug: Nystatin|Drug: Didanosine Argus Pharmaceuticals|NIH AIDS Clinical Trials Information Service Phase 1
    2005-06-23
    NCT00001812 Candidiasis, Oral|Gastrointestinal Diseases|Stomatitis Drug: Nystatin National Cancer Institute (NCI)|National Institutes of Health Clinical Center (CC) Phase 3 1999-04-01 2008-03-03
    NCT00002112 Candidiasis, Oral|HIV Infections Drug: Nystatin|Drug: Fluconazole Pfizer|NIH AIDS Clinical Trials Information Service
    2005-06-23
    NCT01531192 Very Low Birth Weight Infants Dietary Supplement: Lactobacillus reuteri|Drug: Nystatin Zekai Tahir Burak Women's Health Research and Education Hospital Phase 4 2012-06-01 2013-07-13
    NCT00128323 Candidiasis, Oral Drug: Gentian violet 1% solution|Drug: Gentian violet 0.00165% solution|Drug: Nystatin solution University of Malawi College of Medicine|British Society for Antimicrobial Chemotherapy Phase 3 2002-11-01 2008-02-07
    NCT01867164 Vaginitis|Infectious Vaginosis Drug: Gynoclin V|Drug: Vagitrol V Janssen-Cilag, S.A. Phase 3 2007-12-01 2013-11-01
    NCT01718912 Periodontal Disease Drug: metronidazole-nystatin oral rinse Oravital Inc 2013-11-01 2016-03-29
    NCT00002742 Chronic Myeloproliferative Disorders|Infection|Leukemia|Lymphoma|Multiple Myeloma and Plasma Cell Neoplasm|Myelodysplastic Syndromes Drug: amphotericin B deoxycholate|Drug: nystatin Aronex Pharmaceuticals|National Cancer Institute (NCI) Phase 3 1996-01-01 2013-03-25
    NCT01411748 Anticandidal Property of Saccharomyces Boulardii on Very Low Birth Weight Infants Dietary Supplement: Reflor|Drug: mikostatin Zekai Tahir Burak Women's Health Research and Education Hospital Phase 4 2011-07-01 2011-08-05
    NCT01798537 Bacteremia Associated With Intravascular Line|Ventilator Associated Pneumonia|Bacteremia Drug: Neomycin Colistin Nystatin Vancomycin Rambam Health Care Campus Phase 2|Phase 3 2013-06-01 2013-02-25
    NCT00250133 VRE Colonization Procedure: Blood draws University of Pittsburgh Phase 3
    2007-08-31
    NCT02166450 Denture Stomatitis Drug: Nystatin Jagiellonian University 2011-10-01 2014-06-18
    NCT00629122 Kidney Failure, Chronic Drug: Tacrolimus/Clotrimazole Troche|Drug: Tacrolimus/Nystatin Suspension Weill Medical College of Cornell University Phase 4 2008-02-01 2010-11-04

    注:以上所有数据均来自公开文献,并不保证对所有实验均有效,数据仅供参考。

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