Amlodipine是长效的钙离子阻断剂。
Amlodipine is a long-acting calcium channel blocker, used to lower blood pressure and prevent chest pain.
动物 A (mg/kg) = 动物 B (mg/kg)×动物 B的Km系数/动物 A的Km系数 | |
例如,已知某工具药用于小鼠的剂量为88 mg/kg , 则用于大鼠的剂量换算方法:将88 mg/kg 乘以小鼠的Km系数(3),再除以大鼠的Km系数(6),得到该药物用于大鼠的等效剂量44 mg/kg。
[1] Zhang X, et al. Circulation, 1998, 97(6), 576-580.
分子式 C20H25ClN2O5 |
分子量 408.88 |
CAS号 88150-42-9 |
储存方式 ﹣20 ℃冷藏长期储存。冰袋运输 |
溶剂(常温) |
DMSO >25 mg/mL |
Water <1 mg/mL |
Ethanol >25 mg/mL |
体内溶解度
NCT Number | Conditions | Interventions | Sponsor/Collaborators | Phases | Start Date | Last Updated |
NCT02707913 | Healthy | Drug: BF-Amlodipine Tablet 10mg|Drug: Norvasc Tablet 10mg | Bright Future Pharmaceuticals Factory O/B Bright Future Pharmaceutical Laboratories Limited|Chinese University of Hong Kong | Phase 1 | 2016-03-01 | 2016-09-05 |
NCT02064556 | Hypertension | Drug: Amlodipine 10mg|Drug: Amlodipine 10mg/Candesartan 32mg | Chong Kun Dang Pharmaceutical | Phase 1 | 2014-05-01 | 2014-08-13 |
NCT01131936 | Healthy | Drug: Amlodipine | Dr. Reddy's Laboratories Limited | Phase 1 | 2002-08-01 | 2010-06-11 |
NCT01835418 | Hypertension | Drug: Amlodipine | Allina Health System | 2013-04-01 | 2013-04-18 | |
NCT01131923 | Healthy | Drug: Amlodipine | Dr. Reddy's Laboratories Limited | Phase 1 | 2002-10-01 | 2010-06-11 |
NCT00446524 | Hypertension | Drug: Valsartan + Amlodipine besilate | Novartis | Phase 3 | 2007-02-01 | 2012-05-06 |
NCT01356043 | Healthy Male Volunteers | Drug: S-amlodipine 5mg,Telmisartan 80mg|Drug: S-amlodipine 5mg | Chong Kun Dang Pharmaceutical|Asan Medical Center | Phase 1 | 2011-05-01 | 2011-08-29 |
NCT01341392 | Type 2 Diabetes Mellitus | Drug: CKD-501|Drug: amlodiopine|Drug: CKD-501 amlodipine | Chong Kun Dang Pharmaceutical|Severance Hospital | Phase 1 | 2011-04-01 | 2011-08-11 |
NCT01252563 | Hypertension | Drug: Amlodipine | Pfizer | Phase 4 | 2010-12-01 | 2014-01-09 |
NCT02353806 | Chronic Hypertension in Pregnancy | Drug: Amlodipine besylate | University of Texas Southwestern Medical Center|National Center for Advancing Translational Science (NCATS) | Phase 4 | 2015-01-01 | 2016-05-10 |
NCT01278797 | Hypertension | Drug: Telmisartan/Amlodipine Combination Tablet|Drug: Amlodipine Monocomponent | Boehringer Ingelheim | Phase 1 | 2011-01-01 | 2014-02-28 |
NCT01155908 | Healthy | Drug: Amlodipine Besylate / Benazepril Hydrochloride | Dr. Reddy's Laboratories Limited | Phase 1 | 2005-04-01 | 2010-07-01 |
NCT02544776 | Female Infertility Associated With Anovulation | Drug: Clomifene citrate ( clomid 50 mg )|Drug: Amlodipine | Ahmed Fathy Ali Mohamed Ghanem|Ain Shams Maternity Hospital | 2015-01-01 | 2016-03-24 | |
NCT01113047 | Essential Hypertension | Drug: Aliskiren/Amlodipine and Aliskiren/Amlodipine/HCTZ | Novartis | Phase 3 | 2010-05-01 | 2013-12-05 |
NCT01127217 | Hypertension | Drug: amlodipine/losartan|Drug: amlodipine | Hanmi Pharmaceutical Company Limited | Phase 3 | 2009-05-01 | 2010-09-12 |
NCT02974439 | Bioequivalence | Drug: LANDI-Amlodipine Besylate Tablet 5mg|Drug: Norvasc Tablets 5mg | Shanghai Haini Pharmaceutical Co., Ltd. | Phase 1 | 2016-12-01 | 2017-02-13 |
NCT01845272 | Healthy | Drug: candesartan cilexetil 32mg, amlodipine 10mg|Drug: candesartan cilexetil 32mg, amlodipine 10mg | CJ HealthCare Corporation | Phase 1 | 2013-04-01 | 2013-04-30 |
NCT01155895 | Healthy | Drug: Amlodipine Besylate / Benazepril Hydrochloride | Dr. Reddy's Laboratories Limited | Phase 1 | 2004-03-01 | 2010-07-01 |
NCT01926652 | Healthy | Drug: candesartan cilexetil 32mg, amlodipine 10mg | Shin Poong Pharmaceutical Co. Ltd. | Phase 1 | 2013-07-01 | 2013-08-20 |
注:以上所有数据均来自公开文献,并不保证对所有实验均有效,数据仅供参考。
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