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ATP

三磷酸腺苷,Adenosine-Triphosphate,ATP disodium salt

ATP二钠盐是P2嘌呤受体激动剂。

目录号
EY0778
EY0778
EY0778
EY0778
纯度
99.61%
99.61%
99.61%
99.61%
规格
50 mg
100 mg
500 mg
1 g
原价
100
200
300
430
售价
100
200
300
430
库存
现货
现货
现货
现货
订购
订购
订购
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  • 生物活性

    ATP is a disodium salt form of adenosine-triphosphate which is a multifunctional nucleoside triphosphate.

  • 体外研究

  • 体内研究

  • 激酶实验

  • 细胞实验

  • 动物实验

  • 不同实验动物依据体表面积的等效剂量转换表(数据来源于FDA指南)

    动物 A (mg/kg) = 动物 B (mg/kg)×动物 B的Km系数/动物 AKm系数


    例如,已知某工具药用于小鼠的剂量为88 mg/kg , 则用于大鼠的剂量换算方法:将88 mg/kg 乘以小鼠的Km系数(3),再除以大鼠的Km系数(6),得到该药物用于大鼠的等效剂量44 mg/kg。


  • 参考文献

    [1] Chen Y, et al. Science,?006, 314(5806), 1792-1795.
    [2] Guilbert et al (1998) Dependence of P2-nucleotide receptor agonist-mediated endothelium-indepdent relaxation on ectonucleotidase acticity and A2A-receptors in rat portal vein. Br.J.Pharm. 123 1732.
    [3] Burnstock and Kenned (2006) Historical review: ATP as a neurotransmitter. Trends Pharm.Sci. 27 16.
    [4] Gordon (1986) Extracellular ATP: effects, sources and fate. Biochem.J 233 309.

    分子式
    C10H14N5Na2O13P3
    分子量
    551.14
    CAS号
    987-65-5
    储存方式
    ﹣20 ℃冷藏长期储存。冰袋运输
    溶剂(常温)
    DMSO
    <1 mg/mL
    Water
    106 mg/mL
    Ethanol
    <1 mg/mL

    体内溶解度

  • Clinical Trial Information ( data from http://clinicaltrials.gov )

    NCT Number Conditions Interventions Sponsor/Collaborators Phases Start Date Last Updated
    NCT02923726 Sudden Cardiac Death Device: Arm 1 (ATP+Shock)|Device: Arm 2 (shock only) Boston Scientific Corporation|ICON plc 2016-09-01 2016-10-04
    NCT02093611 Muscle Fatigue Caused by Repetitive Muscle Exercise Dietary Supplement: Placebo|Dietary Supplement: ATP Metabolic Technologies Inc.|University of Tampa 2013-07-01 2015-09-24
    NCT02279511 Alzheimer's Disease Drug: ADENOSINE TRIPHOSPHATE|Drug: PLACEBO Sara Varea|Fundacion Clinic per a la Recerca Biom茅dica Phase 2 2014-11-01 2016-05-25
    NCT00147277 Tachycardia, Ventricular|Ventricular Fibrillation Device: Implantable Cardiac Defibrillator Medtronic Bakken Research Center Phase 4 2004-03-01 2015-08-12
    NCT00617578 Ventricular Tachycardia, Monomorphic Device: ATP One Shot ON|Device: ATP One Shot OFF Biotronik SE & Co. KG Phase 4 2007-11-01 2013-12-18
    NCT00147290 Tachycardia, Ventricular|Ventricular Fibrillation Device: Implantable Cardiac Defibrillator Medtronic Bakken Research Center Phase 4 2004-02-01 2015-08-12
    NCT01508338 Healthy Experienced Weight Training Males Dietary Supplement: Placebo|Dietary Supplement: HMB|Dietary Supplement: Peak ATP and HMB|Dietary Supplement: ATP Metabolic Technologies Inc.|University of Tampa 2012-01-01 2014-03-17
    NCT00917696 Osteoarthritis Pain Procedure: Comparator: Iontophoresis and Laser Doppler with ATP|Procedure: Comparator: Iontophoresis and Laser Doppler with Saline Merck Sharp & Dohme Corp. Phase 1 2009-10-01 2015-07-29
    NCT02243631 Calcium Pyrophosphate Deposition Disease Drug: Probenecid VA Office of Research and Development Early Phase 1 2014-10-01 2017-01-04
    NCT02439424 Atrial Tachyarrhythmia|Atrial Fibrillation Device: Reactive ATP Hartford Hospital Phase 1|Phase 2 2015-12-01 2016-12-21
    NCT00565188 Cancer|Palliative Care|Survival|Quality of Life Drug: Adenosine 5'-triphosphate Maastricht University Medical Center|ZonMw: The Netherlands Organisation for Health Research and Development Phase 3 2002-03-01 2016-10-24
    NCT01499069 Overactive Bladder Drug: Oxybutinin, Fesoterodine, Solifenacin, Propiverin, Trospium Samsung Medical Center|Samsung Biomedical Research Institute 2010-02-01 2015-02-12
    NCT00159315 Asthma|COPD|Smoking Procedure: Inhalation Challenge with ATP|Procedure: Inhalation Challenge with AMP Imperial College London|Duska Scientific Co. 2002-10-01 2015-06-03
    NCT01130428 Osteoporosis Device: Juvent 1000 Vibration Platform Maastricht University Medical Center|Research Center for Ageing and Osteoporosis, Copenhagen University Hospital, Copenhagen, Denmark.|University of Sheffield Phase 1|Phase 2 2010-10-01 2011-04-19
    NCT01169246 Ventricular Arrythmias LivaNova|Sorin Group France SAS 2009-11-01 2015-02-23
    NCT00608894 Autoimmune Hepatitis Drug: LCP-Tacro (tacrolimus)|Drug: Azathioprine Veloxis Pharmaceuticals Phase 2 2007-12-01 2014-12-18
    NCT00618267 Multiple Sclerosis Biogen|Elan Pharmaceuticals 2008-03-01 2010-03-04
    NCT01242319 Hypercholesterolemia|Coronary Disease|Primary Health Care|Management, Risk Behavioral: HeartAge intervention Memorial Hospital of Rhode Island|National Heart, Lung, and Blood Institute (NHLBI) 2002-09-01 2010-11-16
    NCT01141504 Healthy Subjects Dietary Supplement: PeakATP 250|Dietary Supplement: Placebo|Dietary Supplement: PeakATP 400|Dietary Supplement: PeakATP 400 plus proprietary blend Metabolic Technologies Inc.|Iowa State University Phase 1 2010-06-01 2012-01-09
    NCT03002038 Neuromyelitis Optica Spectrum Disorder Drug: Azathioprine|Drug: Rituximab Isfahan University of Medical Sciences Phase 2|Phase 3 2015-09-01 2016-12-30
    NCT00098111 Crohn's Disease Drug: azathioprine Massachusetts General Hospital Phase 3 2005-04-01 2014-02-19

    注:以上所有数据均来自公开文献,并不保证对所有实验均有效,数据仅供参考。

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