Sertraline HCl

盐酸舍曲林,CP-51974-1 HCl

Sertraline hydrochloride (盐酸舍曲林) 是选择性5羟色胺再吸收抑制剂(SSRI)。

目录号
EY0513
EY0513
EY0513
EY0513
纯度
99.56%
99.56%
99.56%
99.56%
规格
5 mg
10 mg
25 mg
50 mg
原价
320
480
990
1600
售价
320
480
990
1600
库存
现货
现货
现货
现货
订购
订购
订购
订购
订购
订购
  • 生物活性

    Sertraline HCl is a 5-HT antagonist with Ki of 13 nM.

  • 体外研究

  • 体内研究

  • 激酶实验

  • 细胞实验

  • 动物实验

  • 不同实验动物依据体表面积的等效剂量转换表(数据来源于FDA指南)

    动物 A (mg/kg) = 动物 B (mg/kg)×动物 B的Km系数/动物 AKm系数


    例如,已知某工具药用于小鼠的剂量为88 mg/kg , 则用于大鼠的剂量换算方法:将88 mg/kg 乘以小鼠的Km系数(3),再除以大鼠的Km系数(6),得到该药物用于大鼠的等效剂量44 mg/kg。


  • 参考文献

    [1] Koe BK, et al. J Pharmacol Exp Ther, 1983, 226(3), 686-700.
    [2] Löwe, B., et al. 2005. J Affect Disord. 87: 271-279.
    [3] Khouzam, H.R., et al. 2003. Compr Ther. 29: 47-53.

    分子式
    C17H18Cl3N
    分子量
    342.69
    CAS号
    79559-97-0
    储存方式
    ﹣20 ℃冷藏长期储存。冰袋运输
    溶剂(常温)
    DMSO
    >30 mg/mL
    Water
    <1 mg/mL
    Ethanol
    10 mg/mL

    体内溶解度

  • Clinical Trial Information ( data from http://clinicaltrials.gov )

    NCT01032434 Depression Drug: sertraline Guang Dong Provincial Mental Health Institute 2009-12-01 2015-04-30
    NCT00864019 Healthy Drug: Sertraline HCl 100 mg tablets, single dose|Drug: Zoloft庐 100 mg tablets, single dose Actavis Inc. Phase 1 2004-08-01 2010-08-13
    NCT00969852 Healthy Drug: Sertraline Seoul National University Hospital|Ministry of Health, Welfare and Family Affairs|Korea National Enterprise for Clinical Trials Phase 4 2009-07-01 2011-01-09
    NCT01214382 Roux en Y Gastric Bypass Surgery Drug: Sertraline North Dakota State University|National Institutes of Health (NIH) Phase 3 2010-10-01 2016-04-04
    NCT01267383 Healthy Drug: Sertraline Dr. Reddy's Laboratories Limited Phase 1 2006-09-01 2012-01-10
    NCT01267396 Healthy Drug: Sertraline Dr. Reddy's Laboratories Limited Phase 1 2006-09-01 2012-01-10
    NCT00605813 Depression|Panic Disorder Drug: Sertraline hydrochloride Pfizer 2007-09-01 2012-08-09
    NCT03068429 Obsessive-Compulsive Disorder Drug: Sertraline Hydrochloride University of Sao Paulo Phase 4 2016-12-01 2017-02-24
    NCT02520726 Post-traumatic Stress Disorder Drug: Sertraline University of Utah Phase 4 2013-09-01 2016-10-24
    NCT01802385 Cryptococcal Meningitis|Fungal Meningitis Drug: Sertraline University of Minnesota - Clinical and Translational Science Institute|Infectious Disease Institute, Kampala, Uganda|National Institute of Neurological Disorders and Stroke (NINDS)|Mbarara University of Science and Technology|Ifakara Health Institute Phase 3 2015-03-01 2016-12-06
    NCT01699724 Healthy Drug: JZoloft|Drug: sertraline ODT|Drug: sertraline ODT Pfizer Phase 1 2012-09-01 2012-10-31
    NCT02891278 Acute Myeloid Leukemia Drug: Sertraline|Drug: Cytosine arabinoside|Procedure: allogeneic stem cell transplantation Mark G. Frattini|The Leukemia and Lymphoma Society|Columbia University Phase 1 2016-07-01 2016-09-01
    NCT00605917 Panic Disorder Drug: Sertraline hydrochloride Pfizer 2007-04-01 2012-08-20
    NCT02651623 Healthy Drug: Sertraline|Drug: Moxifloxacin|Drug: Drug - Placebo Pfizer Phase 1 2016-01-01 2016-10-11
    NCT02385799 Autism Spectrum Disorder Drug: Sertraline Liquid Placebo|Drug: Sertraline University of California, Davis|Health Resources and Services Administration (HRSA) Phase 2 2015-02-01 2016-10-24
    NCT02452983 Myelodysplastic Syndromes Drug: Sertraline|Procedure: Bone Marrow Aspirate/Biopsy Gustavo Rivero|Baylor College of Medicine Phase 1 2015-05-01 2017-02-05
    NCT00368550 Alcoholism Drug: Sertraline|Drug: Placebo UConn Health|National Institute on Alcohol Abuse and Alcoholism (NIAAA) Phase 4 2004-02-01 2011-06-17
    NCT01474746 Fragile X Syndrome Drug: Sertraline|Drug: Placebo University of California, Davis Phase 2 2012-01-01 2016-01-26
    NCT00182078 Posttraumatic Stress Disorder|Depression Drug: Placebo|Drug: Sertraline Massachusetts General Hospital Phase 4 2002-11-01 2014-07-08
    NCT01235195 Healthy Drug: sertraline hydrochloride|Drug: sertraline hydrochloride Pfizer Phase 1 2010-11-01 2012-05-17
    NCT01524133 Posttraumatic Stress Disorder Drug: Sertraline|Behavioral: Prolonged Exposure Therapy VA Ann Arbor Healthcare System|U.S. Army Medical Research and Materiel Command Phase 4 2011-11-01 2016-06-16

    注:以上所有数据均来自公开文献,并不保证对所有实验均有效,数据仅供参考。

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