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Lapatinib Ditosylate is the xylenesulfonic acid salt form of lapatinib (GW-572016), a small-molecule dual inhibitor of EGFR and ErbB2 receptor kinase activities. Lapatinib ditosylate (甲苯磺酸拉帕替尼; GW-572016 ditosylate) 是EGFR和ErbB2抑制剂，IC50分别为10.8和9.2 nM。
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(+)-JQ1, an active enantiomer of JQ1, is a potent, highly specific and Kac-competitive inhibitor of bromodomain and extraterminal domain (BET) proteins, blocks BRD4 resulting in inhibition of c-Myc expression and tumor growth. (+)-JQ1是一种BET bromodomain抑制剂，作用于BRD4(2)，IC50为33 nM，结合到BET家族的所有Bromodomain结构域，而不结合到BET家族以外的Bromodomain结构域。
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Ricolinostat (ACY-1215) is an oral, first-in-class, selective inhibitor of HDAC6, and inhibits tubulin deacetylase. Rocilinostat (ACY-1215)是高效HDAC6抑制剂，IC50为5 nM，比对HDAC1/2/3的抑制性高10倍以上，对HDAC8有微弱活性，对HDAC4/5/7/9/11，Sirtuin1和Sirtuin2活性最低。
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Kartogenin (KGN), a small molecular compound, can induce bone marrow-derived mesenchymal stem cells (BMSCs) into chondrocytes. Kartogenin是针对软骨形成的小分子激动剂，促进软骨细胞分化（EC50为100nM），结合filamin A，并阻止其与转录因子CBFβ)的相互作用。
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KX2-391 (KX-01), the first peptidomimetic Src kinase inhibitor, is a synthetic, orally bioavailable inhibitor that has tubulin polymerization inhibition as a second mechanism of action, and is currently in Phase-2 testing for solid tumors. KX2-391 (KX01)是第一个进入临床的拟肽类Src抑制剂，靶向Src的多肽底物结合位点，对多种癌细胞株GI50为9-60 nM。
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