MCT
MCTs (The monocarboxylate transporters) are a family of proton-linked plasma membrane transporters that carry molecules having one carboxylate group (monocarboxylates), such as lactate and pyruvate, across biological membranes.
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Olaparib (AZD2281, Ku-0059436)是一种选择性的PARP1/2抑制剂，IC50为5 nM/1 nM，比对Tankyrase-1的抑制作用强300倍。
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KN-93 H3PO4 是一种强效的特异性的Ca2+/calmodulin-dependent protein kinase II (CaMKII)抑制剂，其 Ki 为 0.37 μM,对 APK, PKC, MLCK 或 Ca2+-PDE 没有明显的抑制活性。
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BAPTA-AM 是选择透过性膜calcium螯合剂。
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Tranylcypromine hydrochloride is a racemic mixture of (±)-Trans-2-phenylcyclopropyl-1-amine (TCP, tPCPA) · HCl that covalently inhibits the LSD and MAO enzymes. Tranylcypromine (2-PCPA) HCl是一种非选择性的不可逆的单胺氧化酶(MAO)抑制剂，用作抗抑郁药和抗焦虑药。
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Iniparib (BSI-201)是一种PARP1抑制剂，对三阴性乳腺癌(TNBC)有效。
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