Fulvestrant是一种Estrogen receptor(ER)(雌激素受体)拮抗剂, IC50为0.094 nM。
MoreTamoxifen citrate, a selective non-steroidal estrogen receptor antagonist, was approved by FDA as a drug that is utilized in the treatment of estrogen receptor–positive breast cancer. Tamoxifen Citrate是一种雌激素受体拮抗剂,与雌激素竞争性结合。
MoreEquol是是大豆的代谢物,是人类的一种重要的异黄酮,与5α-DHT特异性结合,对重组雌激素受体ERβ具有适度的亲和力。
MoreOspemifene is a non-hormonal selective estrogen receptor modulator (SERM) which is used for the treatment of dyspareunia.
MoreEthisterone为可作用于前列腺癌的孕激素。
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