Adrenergic Receptor
The adrenergic receptors (or adrenoceptors) are a class of G protein-coupled receptors that are targets of the catecholamines, especially norepinephrine (noradrenaline) and epinephrine (adrenaline). Epinephrine (adrenaline) reacts with both α- and β-adrenoreceptors, causing vasoconstriction and vasodilation, respectively. High levels of circulating epinephrine cause vasoconstriction. At lower levels of circulating epinephrine, β-adrenoreceptor stimulation dominates, producing vasodilation followed by decrease of peripheral vascular resistance.
Many cells possess these receptors, and the binding of a catecholamine to the receptor will generally stimulate the sympathetic nervous system. The sympathetic nervous system is responsible for the fight-or-flight response, which includes dilating the pupils, increasing heart rate, mobilizing energy, and diverting blood flow from non-essential organs to skeletal muscle.
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BRL 44408 maleate是选择性 α2A 拮抗剂。
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BRL 37344， sodium salt是β3 激动剂。
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BMY 7378 dihydrochloride是选择性 α1D 拮抗剂。
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B-HT 933 dihydrochloride是选择性 α2 激动剂。
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B-HT 920是D2 受体激动剂。 也是 α2 激动剂，5-HT3 拮抗剂。
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BRL 44408 maleate是选择性 α2A 拮抗剂。
More
-
BRL 37344， sodium salt是β3 激动剂。
More
-
BMY 7378 dihydrochloride是选择性 α1D 拮抗剂。
More
-
B-HT 933 dihydrochloride是选择性 α2 激动剂。
More
-
B-HT 920是D2 受体激动剂。 也是 α2 激动剂，5-HT3 拮抗剂。
More
