T0070907 (T007), a potent and selective PPARγ inhibitor, can reduce α and β tubulin proteins in some cancer cell lines. T0070907是一种选择性的PPARγ抑制剂,IC50为1 nM,比作用于PPARα和PPARδ选择性高800倍以上。
MoreWY-14643 (Pirinixic Acid), a moderate dual PPARα/γ activator, inhibits neuroinflammation and oxidative stress, and also possesses antidepressive activities. WY-14643 (Pirinixic Acid)是一种有效的过氧化物酶体增殖子和PPARα激活剂,EC50为1.5 μM。
MoreGSK3787 is a selective and irreversible PPARβ/δ antagonist with good pharmacokinetic properties. GSK3787是不可逆的PPARδ选择性拮抗剂,pIC50为6.6,对hPPARα和hPPARγ无亲和力。
MoreNaringenin, a common dietary flavonoid abundantly present in fruits and vegetables, is believed to possess strong anti-proliferative properties and the ability to induce apoptosis in hepatoma cell lines.
MoreClofibric Acid是PPARα激动剂,是一种降血脂剂。
MoreT0070907 (T007), a potent and selective PPARγ inhibitor, can reduce α and β tubulin proteins in some cancer cell lines. T0070907是一种选择性的PPARγ抑制剂,IC50为1 nM,比作用于PPARα和PPARδ选择性高800倍以上。
MoreWY-14643 (Pirinixic Acid), a moderate dual PPARα/γ activator, inhibits neuroinflammation and oxidative stress, and also possesses antidepressive activities. WY-14643 (Pirinixic Acid)是一种有效的过氧化物酶体增殖子和PPARα激活剂,EC50为1.5 μM。
MoreGSK3787 is a selective and irreversible PPARβ/δ antagonist with good pharmacokinetic properties. GSK3787是不可逆的PPARδ选择性拮抗剂,pIC50为6.6,对hPPARα和hPPARγ无亲和力。
MoreNaringenin, a common dietary flavonoid abundantly present in fruits and vegetables, is believed to possess strong anti-proliferative properties and the ability to induce apoptosis in hepatoma cell lines.
MoreClofibric Acid是PPARα激动剂,是一种降血脂剂。
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