GABA Receptor
GABA receptors are a class of receptors that respond to the neurotransmitter gamma-aminobutyric acid (GABA), the chief inhibitory compound in the mature vertebrate central nervous system. GABA receptors influence cognition by coordinating with glutamatergic processes. There are two classes of GABA receptors: GABAA and GABAB. GABAA receptors are ligand-gated ion channels; whereas GABAB receptors are G protein-coupled receptors, also called metabotropic receptors. A subclass of ionotropic GABA receptors, insensitive to typical allosteric modulators of GABAA receptor channels such as benzodiazepines and barbiturates, designated GABAС receptor.
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Rosuvastatin Calcium是一种竞争性HMG-CoA还原酶抑制剂， with IC50为11 nM。
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(R)-baclofen是一种γ-氨基丁酸衍生物，主要用于治疗痉挛。是选择性GABAB受体激动剂。
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KU-0060648是DNA-PK和PI3Kα/β/δ双重抑制剂，IC50分别为8.6 nM和4 nM/0.5 nM/0.1 nM，对PI3Kγ抑制作用稍弱，IC50为0.59 μM。
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Baicalin is a known prolyl endopeptidase inhibitor that induces apoptosis in pancreatic cancer cells.
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Clinofibrate抑制hydroxymethylglutaryl coenzyme A reductase (HMGCR)（羟甲基戊二酰辅酶A还原酶），IC50为0.47 mM，是一种降脂剂，用于控制血液中的高胆固醇和甘油三酯水平。
More
-
Rosuvastatin Calcium是一种竞争性HMG-CoA还原酶抑制剂， with IC50为11 nM。
More
-
(R)-baclofen是一种γ-氨基丁酸衍生物，主要用于治疗痉挛。是选择性GABAB受体激动剂。
More
-
KU-0060648是DNA-PK和PI3Kα/β/δ双重抑制剂，IC50分别为8.6 nM和4 nM/0.5 nM/0.1 nM，对PI3Kγ抑制作用稍弱，IC50为0.59 μM。
More
-
Baicalin is a known prolyl endopeptidase inhibitor that induces apoptosis in pancreatic cancer cells.
More
-
Clinofibrate抑制hydroxymethylglutaryl coenzyme A reductase (HMGCR)（羟甲基戊二酰辅酶A还原酶），IC50为0.47 mM，是一种降脂剂，用于控制血液中的高胆固醇和甘油三酯水平。
More
