Cannabinoid Receptor
Cannabinoid receptors, located throughout the body, are part of the Endocannabinoid system which is involved in a variety of physiological processes including appetite, pain-sensation, mood, and memory.
Cannabinoid receptors are of a class of cell membrane receptors under the G protein-coupled receptor superfamily. As is typical of G protein-coupled receptors, the cannabinoid receptors contain seven transmembrane spanning domains. Cannabinoid receptors are activated by three major groups of ligands: endocannabinoids, produced by the mammillary body; plant cannabinoids; and synthetic cannabinoids. There are currently two known subtypes of cannabinoid receptors, termed CB1 and CB2.
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Bay 59-3074是CB1/CB2 受体 部分 激动剂。
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Arvanil是活性的 CB1 和 TRPV1 激动剂。 也是anandamide 转运抑制剂。
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AM 6545是高亲和性，选择性 CB1 拮抗剂。
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AM 281是活性的，选择性 CB1 拮抗剂/反相激动剂。
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Abn-CBD是选择性 GPR55 激动剂， 神经行为性失活。
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