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Rivastigmine tartrate (酒石酸卡巴拉汀) 是胆碱酯酶抑制剂，IC50为5.5 uM，还能抑制丁酰胆碱酯酶和乙酰胆碱酯酶。
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PHT-427是作用于Akt和PDPK1的双重抑制剂，Akt和PDPK1的PH结构域具有高度亲和力，Ki分别为2.7 μM和5.2 μM。
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Laetrile is a glycoside initially isolated from the seeds of the tree Prunus dulcis, also known as bitter almonds.Amygdalin isolated from S. Persicae extract in ISF-1 through a bioactivity-guided fractionation procedure induced the expression of follistatin in HepG2 and C2C12 cell lines.The amygdalin induced increase in TCCSUP migratory behavior indicates that any anti-tumor benefits from amygdalin (seen with the other two cell lines) may depend upon the cancer cell type.Amygdalin is a natural product that owns antitumor activity, less side effects, widely sourced and relatively low priced.
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Zafirlukast (扎鲁司特) 是口服活性的白三烯受体拮抗剂（LTRA）。
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Raltegravir是一种有效的整合酶链转移抑制剂，作用于WT和S217Q原型泡沫病毒(PFV)整合酶，IC50分别为90 nM和40 nM。
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