Ivermectin是广谱的抗寄生虫化合物,是α7神经元烟碱乙酰胆碱受体和P2X4受体阳性变构调节剂。
MoreSpectinomycin双盐酸盐是不经肠道的抗生素,由壮观链霉菌制备而来。Spectinomycin hydrochloride is a new parenteral antibiotic prepared from Streptomyces spectabilis. Spectinomycin (hydrochloride) is structurally related to aminoglycosides. Spectinomycin lacks amino sugar and glycosidic bonds. Spectinomycin has moderate antibacterial activity against many gram positive and gram negative bacteria but Spectinomycin (hydrochloride) is especially effective against Niesseria gonorrhoeae.
MoreAnacardic Acid是一个有效的p300 and p300/CBP-associated factor histone acetyltranferases的抑制剂,也具有抗细菌和抗微生物活性,抑制前列腺素合成,并抑制酪氨酸酶和脂肪氧合酶。
MoreDabigatran etexilate是口服活性的dabigatran原药,是可逆的直接凝血酶抑制剂(DTI),Ki为4.5 nM。
More20-Hydroxyecdysone是一种自然发生的蜕皮激素,控制节肢动物的蜕皮和变态。
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