VO-OHpic trihydrate是PTEN(phosphatase and tensin homologue deleted on chromosome 10)高活性抑制剂,IC50值为35 nM。
MoreFirategrast是口服有效的整合素α4β1/α4β7小分子拮抗剂。
MoreFAK Inhibitor 14 is a selective focal adhesion kinase (FAK) inhibitor, it prevents FAK autophosphorylation at Y397 (IC50 = 1μM).
MoreMyD88的二聚化抑制剂。
MoreCP-640186 hydrochloride是乙酰辅酶A羧化酶(ACCase)抑制剂,对鼠肝ACCase1和骨骼肌ACCase2的IC50s分别为53 nM和61 nM。
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