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Other Singal pathway


  • Nutlin-3a EY0963

    Nutlin-3a是Nutlin-3的活性对映体,抑制p53/MDM2相互作用,IC50为90 nM。

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  • Temsirolimus EY0969

    Temsirolimus (CCI-779) is a specific mTOR inhibitor with IC50 of 1.76 μM。

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  • WP1066 EY0931

    WP1066是一种新型JAK2和STAT3抑制剂,IC50分别为2.30 μM和2.43 μM;对JAK2, STAT3, STAT5和ERK1/2具有抑制活性,但不抑制JAK1和JAK3。

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  • Dimethyloxallyl Glycine EY0946

    Dimethyloxallyl Glycine(DMOG)是可渗透入细胞的HIF-1α脯氨酰羟化酶(HIF-PH)竞争性抑制剂。

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  • Fasudil HCl EY0908

    Fasudil (HA-1077) HCl是一种有效的ROCK-II, PKA, PKG, PKC,和MLCK抑制剂, Ki分别为0.33 μM, 1.6 μM, 1.6 μM, 3.3 μM,和36 μM。

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