MK-8745是一种高度选择性Aurora-A抑制剂,IC50 为0.6 nM,其对于Aurora-A的选择性高于Aurora B的选择性450倍。
MoreSNS-032是CDK 9,2和7的抑制剂,IC50分别为4,38和62 nM。
MorePelitinib (EKB-569; WAY-EKB 569)是不可逆的EGFR抑制剂,IC50为38.5 nM。
MoreBaicalin is a known prolyl endopeptidase inhibitor that induces apoptosis in pancreatic cancer cells.
MorePF-431396 is dual focal adhesion kinase (FAK) and proline-rich tyrosine kinase 2 (PYK2) inhibitor (IC50 values are 2 and 11 nM respectively), PF-431396 has a Kd value of 445 nM for BRD4.
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