Pelitinib (EKB-569; WAY-EKB 569)是不可逆的EGFR抑制剂,IC50为38.5 nM。
MoreBaicalin is a known prolyl endopeptidase inhibitor that induces apoptosis in pancreatic cancer cells.
MorePF-431396 is dual focal adhesion kinase (FAK) and proline-rich tyrosine kinase 2 (PYK2) inhibitor (IC50 values are 2 and 11 nM respectively), PF-431396 has a Kd value of 445 nM for BRD4.
MoreValdecoxib是一种强有效和选择性的COX-2抑制剂,IC50为5nM.
MoreEstradiol cypionate是一种合成酯,是长效雌激素。
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