Naringenin, a common dietary flavonoid abundantly present in fruits and vegetables, is believed to possess strong anti-proliferative properties and the ability to induce apoptosis in hepatoma cell lines.
MoreLY2874455能抑制FGF/FGFR介导的信号转导,有广谱抗癌活性。
MorePiceatannol,是一种天然二苯乙烯,是选择性Syk抑制剂,比作用于Lyn选择性高10倍左右。
MoreAZ20是高活性ATR抑制剂,IC50为5 nM,对mTOR的IC50为38 nM。
MoreLDN-57444是一种可逆的竞争性的蛋白酶体抑制剂,,抑制UCch-L1时,IC50为0.88 μM,比作用于亚型Uch-L3选择性高30倍。
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