EGF816 is a third-generation covalent EGFR inhibitor that has potent inhibitory activity against activating and resistant T790M mutants with low IC50 in various cellular assays.
MoreHM-71224 is an EGFR tyrosine kinase inhibitor.
MoreAvosentan是内皮素(ETA)受体拮抗剂。
MoreSuvorexant是OX受体拮抗剂,对OX1和OX2受体的Ki分别为0.55 nM和0.35 nM。
MoreBoceprevir是HCV蛋白酶抑制剂,Ki为14 nM。
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