Procaine is an inhibitor of sodium channel, NMDA receptor and nAChR with IC50 of 60 μM, 0.296 mM and 45.5 μM, which is also an inhibitor of 5-HT3 with KD of 1.7 μM.
MoreHomatropine Methylbromide is muscarinic AChR antagonist, inhibits endothelial and smooth muscle muscarinic receptors of WKY-E and SHR-E with IC50 of 162.5 nM and 170.3 nM, respectively.
MoreBetahistine is a histamine H3 receptor inhibitor with IC50 of 1.9 μM.
MoreBrinzolamide is a potent carbonic anhydrase II inhibitor with IC50 of 3.19 nM.
MoreFlumequine is a synthetic chemotherapeutic antibiotic, inhibiting topoisomerase II with IC50 of 15 μM.
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