Rucaparib phosphate是PARP抑制剂,对PARP1的Ki为1.4 nM,对PARP其余亚型也有亲和性。
MoreSU11274(PKI-SU11274)是Met抑制剂,IC50为10 nM,对PGDFRβ,EGFR和Tie2无活性。
MoreGSK J4 hydrochloride is a cell permeable prodrug of GSK J1, which is the first selective inhibitor of the H3K27 histone demethylase JMJD3 and UTX with IC50 of 60 nM and inactive against a panel of demethylases of the JMJ family.
MoreBleomycin Sulfate是一种糖肽类抗生素,作用于UT-SCC-19A细胞,IC50为4 nM。
MoreLY2228820是p38MAPK抑制剂,对p38αMAPK和p38βMAPK的IC50分别为7 nM和3 nM。
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